SCHEMBL3045890

SCHEMBL3045890

O=CC(=O)c1ccc(Br)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
MAPK1 P28482 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
CES2 O00748 1/20 0.56
CES1 P23141 1/20 0.56
RAB9A P51151 2/20 0.53
LMNA P02545 2/20 0.53
RECQL P46063 1/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
MAPT P10636 3/20 0.52
CYP1B1 Q16678 1/20 0.52
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
GSK3B P49841 2/20 0.48
CYP1A2 P05177 1/20 0.47
OGG1 O15527 1/20 0.46
NPC1 O15118 1/20 0.46
AKR1C3 P42330 1/20 0.45
HDAC3 O15379 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL28480633 0.98 ALDH1A1 (0.56) ALDH1A1MAPK1TDP1CES2CES1
SCHEMBL222221 0.87 ALDH1A1 (0.74) ALDH1A1MAPK1TDP1RAB9ALMNA
Water SCHEMBL11592742 0.84 ALDH1A1 (0.70) ALDH1A1MAPK1TDP1RAB9ALMNA
Water SCHEMBL11592745 0.84 ALDH1A1 (0.70) ALDH1A1MAPK1TDP1RAB9ALMNA
SCHEMBL8586818 0.82 RAB9A (0.67) ALDH1A1TDP1CES2CES1RAB9A
SCHEMBL8586821 0.82 RAB9A (0.67) ALDH1A1TDP1CES2CES1RAB9A
Xenygloxal SCHEMBL2110325 0.79 ALDH1A1 (0.64) ALDH1A1MAPK1TDP1RAB9ALMNA
SCHEMBL11530261 0.79 ALDH1A1 (0.64) ALDH1A1MAPK1TDP1RAB9ALMNA
SCHEMBL28128609 0.79 ALDH1A1 (0.46) ALDH1A1MAPK1TDP1CES2CES1
SCHEMBL8864790 0.78 ALDH5A1 (0.64) ALDH1A1MAPK1TDP1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 83 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117417248-A Molecular-level monolayer hydrophilic graphene quantum dot and preparation method thereof 武汉科技大学 2024-01-19 CN claimed
CN-115947911-B Diketimine-linked covalent organic framework polymer material and preparation method thereof 天津大学 2023-05-23 CN claimed
CN-115947911-A Diketimine-linked covalent organic framework high polymer material and preparation method thereof 天津大学 2023-04-11 CN claimed
CN-113512073-A Synthesis of novel non-doped nickel-based metal organic complex hole transport material and application of novel non-doped nickel-based metal organic complex hole transport material in perovskite type solar cell 云南大学 2021-10-19 CN claimed
US-12195450-B2 Small molecule neutral sphingomyelinase 2 (nSMase2) inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2025-01-14 US disclosed
WO-2024249950-A1 FUSED PYRIMIDINE COMPOUNDS AS INHIBITORS OF MENIN BIOMEA FUSION, INC. (US) 2024-12-05 WO disclosed
CN-118994018-A Synthesis method of 1,3, 4-triarylimidazole thioketone derivative 江苏建筑职业技术学院 2024-11-22 CN disclosed
CN-115521196-B Method for preparing alpha-hydroxy ketone compound by using water as hydrogen source 云南民族大学 2024-03-29 CN disclosed
CN-117510478-A Design, synthesis and application of organic photocatalyst based on pyrazine and quinoxaline skeleton 瑞博(苏州)制药有限公司 2024-02-06 CN disclosed
CN-117417248-A Molecular-level monolayer hydrophilic graphene quantum dot and preparation method thereof 武汉科技大学 2024-01-19 CN disclosed
CN-115504946-B Method for synthesizing alpha-ketoamide compound 武汉工程大学 2023-12-15 CN disclosed
CN-111995591-B Dicyanopyrazine compound, light-emitting material, and light-emitting element using same 国立大学法人九州大学 2023-12-08 CN disclosed
US-20050075340-A1 Triazolotriazine compounds and uses thereof SUGEN, INC. 2005-04-07 US disclosed
WO-2005010005-A1 TRIAZOLOTRIAZINE COMPOUNDS AND USES THEREOF SUGEN, INC. (US) 2005-02-03 WO disclosed
WO-2003052053-A2 NUCLEOSIDE LIBRARIES AND COMPOUNDS BY MCC COMBINATORIAL STRATEGIES ON SOLID SUPPORT RIBAPHARM INC. (US) 2003-06-26 WO disclosed
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US disclosed
CN-1349514-A Triazine derivatives having insecticidal activity SINGENTA PARTICIPATION AG (CH) 2002-05-15 CN disclosed
US-4071570-A ANTIARRHYTHMIC AGENTS MERCK & CO., INC. (US) 1978-01-31 US disclosed
US-3978127-A ANTIARRHYTHMIC MERCK & CO., INC. (US) 1976-08-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12195450-B2 Small molecule neutral sphingomyelinase 2 (nSMase2) inhibitors SMPD2, SPTLC2, SGMS2 ALDH1A1 3995/4885MAPK1 1963/4885TDP1 826/4885
US-20050075340-A1 Triazolotriazine compounds and uses thereof MET, TPMT, RET ALDH1A1 439/4885MAPK1 2029/4885TDP1 3239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.