SCHEMBL30488585

SCHEMBL30488585

COc1ccc2c(c1)OCC(N)=C2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.55
NR1H4 Q96RI1 2/20 0.50
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
KDM4E B2RXH2 5/20 0.40
MAPT P10636 5/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
ALDH1A1 P00352 4/20 0.40
CYP3A4 P08684 2/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MTNR1A P48039 2/20 0.40
CA2 P00918 1/20 0.40
CA5A P35218 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9729530 0.76 ALOX5 (0.54) ALOX5NR1H4CA12CA9KDM4E
SCHEMBL31544361 0.76 ALOX5 (0.54) ALOX5NR1H4CA12CA9KDM4E
SCHEMBL430257 0.76 ALOX5 (0.51) ALOX5NR1H4CA12CA9KDM4E
SCHEMBL10470600 0.75 ALOX5 (0.71) ALOX5NR1H4CA12CA9MAPT
SCHEMBL432850 0.75 ALOX5 (0.71) ALOX5NR1H4CA12CA9KDM4E
SCHEMBL10702114 0.73 ALOX5 (0.57) ALOX5NR1H4CA12CA9KDM4E
SCHEMBL30438234 0.73 ALOX5 (0.48) ALOX5NR1H4CA12CA9KDM4E
SCHEMBL7058640 0.73 PTGS2 (0.51) ALOX5NR1H4KDM4EMAPTSMN1; SMN2
SCHEMBL18055910 0.72 ALOX5 (0.53) ALOX5NR1H4CA12CA9KDM4E
Formamide SCHEMBL9729804 0.71 MTNR1A (0.56) ALOX5NR1H4CA12CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478143-A Donepezil derivative, preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2023-07-25 CN claimed
CN-116478143-A Donepezil derivative, preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2023-07-25 CN disclosed