SCHEMBL30516400

SCHEMBL30516400

[2H]c1c([2H])c([2H])c(-c2c(C(=O)O)ccn2S(=O)(=O)c2cccnc2)c(F)c1[2H]

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
HTT P42858 2/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
NAPRT Q6XQN6 1/20 0.35
POLB P06746 1/20 0.34
ALDH1A1 P00352 3/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
SLC6A9 P48067 1/20 0.33
PIK3CG P48736 1/20 0.33
FABP4 P15090 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30516399 1.00 KDM4E (0.38) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30516378 0.82 ERN1 (0.33) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30516401 0.78 KDM4E (0.37) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL29051062 0.78 KDM4E (0.37) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL28649101 0.75 CHRNB2 (0.41) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30267526 0.75 CHRNB2 (0.41) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL28695918 0.74 KDM4E (0.46) KDM4ENAPRTPOLBALDH1A1HPGD
SCHEMBL30516405 0.71 NFE2L2 (0.33) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL30748189 0.71 TP53 (0.40) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL29141637 0.71 TP53 (0.40) KDM4ECHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108794449-B Synthetic method of deuterated fumaric acid vorofacian metabolite 广东东阳光药业有限公司 2023-08-04 CN claimed
CN-108794449-B Synthetic method of deuterated fumaric acid vorofacian metabolite 广东东阳光药业有限公司 2023-08-04 CN disclosed