SCHEMBL30516378

SCHEMBL30516378

[2H]c1c([2H])c([2H])c(-c2c(C=O)ccn2S(=O)(=O)c2cccnc2)c(F)c1[2H]

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.33
NAPRT Q6XQN6 1/20 0.33
CYP2C19 P33261 1/20 0.32
HTT P42858 2/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
KDM4E B2RXH2 1/20 0.32
FGFR4 P22455 1/20 0.31
POLB P06746 1/20 0.31
SLC40A1 Q9NP59 1/20 0.30
CYP17A1 P05093 1/20 0.30
CYP21A2 P08686 1/20 0.30
CYP11B1 P15538 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
MET P08581 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28558398 0.84 CHRNB2 (0.38) ERN1NAPRTCYP2C19HTTCHRNB2
SCHEMBL29538386 0.84 CHRNB2 (0.38) ERN1NAPRTCYP2C19HTTCHRNB2
SCHEMBL30516400 0.82 KDM4E (0.38) NAPRTHTTCHRNB2CHRNB4CHRNA3
SCHEMBL30516399 0.82 KDM4E (0.38) NAPRTHTTCHRNB2CHRNB4CHRNA3
SCHEMBL30516405 0.78 NFE2L2 (0.33) ERN1NAPRTHTTCHRNB2CHRNB4
SCHEMBL30544721 0.78 NAPRT (0.41) ERN1NAPRTCYP2C19CHRNB2CHRNB4
SCHEMBL1156745 0.74 NAPRT (0.42) NAPRTCYP2C19KDM4EFGFR4MET
SCHEMBL28512380 0.73 NAPRT (0.41) ERN1NAPRTCYP2C19KDM4EFGFR4
SCHEMBL30516401 0.71 KDM4E (0.37) NAPRTHTTCHRNB2CHRNB4CHRNA3
SCHEMBL29051062 0.71 KDM4E (0.37) NAPRTHTTCHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108794449-B Synthetic method of deuterated fumaric acid vorofacian metabolite 广东东阳光药业有限公司 2023-08-04 CN claimed
CN-108794449-B Synthetic method of deuterated fumaric acid vorofacian metabolite 广东东阳光药业有限公司 2023-08-04 CN disclosed
CN-108794449-B Synthetic method of deuterated fumaric acid vorofacian metabolite 广东东阳光药业有限公司 2023-08-04 CN disclosed