SCHEMBL305837

SCHEMBL305837

CON(C)C(=O)c1cccc(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.53
CES1 P23141 2/20 0.53
TRPM8 Q7Z2W7 1/20 0.51
PARP1 P09874 1/20 0.50
OPRM1 P35372 1/20 0.49
OPRL1 P41146 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
TSHR P16473 1/20 0.48
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.48
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
LMNA P02545 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MLYCD O95822 1/20 0.46
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GRM1 Q13255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29729945 1.00 CES2 (0.53) CES2CES1TRPM8PARP1OPRM1
SCHEMBL14784157 0.91 TRPM8 (0.56) CES2CES1TRPM8OPRM1OPRL1
SCHEMBL30678242 0.88 NPC1 (0.49) CES2CES1TRPM8OPRM1OPRL1
SCHEMBL15281239 0.87 KMT2A (0.50) CES2CES1TRPM8PARP1TSHR
SCHEMBL906184 0.84 CES2 (0.55) CES2CES1PARP1OPRM1OPRL1
SCHEMBL16214051 0.82 MEN1 (0.46) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL255000 0.82 CES2 (0.61) CES2CES1PARP1OPRM1OPRL1
SCHEMBL3651911 0.82 MLYCD (0.47) CES2CES1TRPM8NPC1RAB9A
SCHEMBL29482201 0.82 CES2 (0.61) CES2CES1PARP1OPRM1OPRL1
SCHEMBL2652369 0.81 HPGD (0.57) PARP1NPC1RAB9AHDAC6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 264 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12534457-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2026-01-27 US disclosed
US-12528799-B2 Heteroaryl derivative compounds, and uses thereof VORONOI INC. (KR) 2026-01-20 US disclosed
US-20250368635-A1 HETEROARYL DERIVATIVE COMPOUND, AND USES THEREOF VORONOI, INC. (KR) 2025-12-04 US disclosed
EP-4631507-A2 HETEROARYL DERIVATIVE, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS EFFECTIVE COMPONENT Voronoi Inc. (KR) 2025-10-15 EP disclosed
EP-4619403-A1 HETEROARYL DERIVATIVE COMPOUND, AND USES THEREOF Voronoi, Inc. (KR) 2025-09-24 EP disclosed
EP-3943491-B1 HETEROARYL DERIVATIVE, METHOD FOR PRODUCING SAME, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS EFFECTIVE COMPONENT VORONOI INC (KR) 2025-06-18 EP disclosed
US-20250019373-A1 ARYL OR HETEROARYL DERIVATIVE, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF KINASE-RELATED DISEASES VORONOI INC. (KR) 2025-01-16 US disclosed
US-12157730-B2 Heteroaryl derivative, method for producing same, and pharmaceutical composition comprising same as effective component VORONOI INC. (KR) 2024-12-03 US disclosed
US-12152021-B2 Heteroaryl derivative, method for producing same, and pharmaceutical composition comprising same as effective component VORONOI INC. (KR) 2024-11-26 US disclosed
US-20240317730-A1 HETEROARYL DERIVATIVE COMPOUNDS, AND USES THEREOF VORONOI INC. (KR) 2024-09-26 US disclosed
WO-2004052868-A1 PYRAZINE-BASED TUBULIN INHIBITORS CYTOPIA PTY LTD (AU) 2004-06-24 WO disclosed
WO-2004043458-A1 BICYCLIC-SUBSTITUTED AMINES AS HISTAMINE-3 RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2004-05-27 WO disclosed
US-20040092521-A1 Bicyclic-substituted amines as histamine-3 receptor ligands ABBOTT LABORATORIES 2004-05-13 US disclosed
EP-1115729-A1 PHOSPHONIC ACID DERIVATIVES AS INHIBITORS OF PTP-1B Merck Frosst Canada & Co. (CA) 2001-07-18 EP disclosed
US-6174874-B1 ANTIDIABETIC,-CARCINOGENIC AGENTS; IMPROVING GLUCOSE TOLERANCE/INSULIN-SENSITIVITY; PREVENTING/TREATING OBESITY AND NEURODEGENERATIVE DISEASES; E.G. 1,3-BIS-((PHOSPHONODI-FLUOROMETHYL)PHENYL)-2-DICARBOXYPROPANE MERCK FROSST CANADA & CO. (CA) 2001-01-16 US disclosed
EP-1031572-A1 PYRIDYLPYRROLE DERIVATIVES Sankyo Company Limited (JP) 2000-08-30 EP disclosed
WO-2000017211-A1 PHOSPHONIC ACIDS DERIVATIVES AS INHIBITORS OF PTP-1B MERCK FROSST CANADA & CO. (CA) 2000-03-30 WO disclosed
US-5494918-A ANTICHOLESTEROL AGENTS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-02-27 US disclosed
US-5385912-A Hypocholesterolemic or hypolipidemic agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1995-01-31 US disclosed
WO-1992015579-A1 MULTICYCLIC TERTIARY AMINE POLYAROMATIC SQUALENE SYNTHETASE INHIBITORS RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1992-09-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12157730-B2 Heteroaryl derivative, method for producing same, and pharmaceutical composition comprising same as effective component ERBB4, ERBB2, EGFR CES2 3680/4885CES1 3409/4885TRPM8 2466/4885
US-20250368635-A1 HETEROARYL DERIVATIVE COMPOUND, AND USES THEREOF ERBB2, EGFR, ERBB3 CES2 2512/4885CES1 3354/4885TRPM8 2519/4885
US-12152021-B2 Heteroaryl derivative, method for producing same, and pharmaceutical composition comprising same as effective component ERBB4, ERBB2, EGFR CES2 3680/4885CES1 3409/4885TRPM8 2466/4885
US-20240317730-A1 HETEROARYL DERIVATIVE COMPOUNDS, AND USES THEREOF ERBB2, EGFR, ERBB3 CES2 2857/4885CES1 3727/4885TRPM8 3409/4885
US-12528799-B2 Heteroaryl derivative compounds, and uses thereof ERBB2, EGFR, ERBB3 CES2 1116/4885CES1 706/4885TRPM8 2503/4885
US-12534457-B2 Heteroaryl derivative compounds, and uses thereof ERBB2, EGFR, ERBB3 CES2 1186/4885CES1 807/4885TRPM8 856/4885
US-20040092521-A1 Bicyclic-substituted amines as histamine-3 receptor ligands HRH3, HRH4, HRH1 CES2 1258/4885CES1 827/4885TRPM8 377/4885
US-20250019373-A1 ARYL OR HETEROARYL DERIVATIVE, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF KINASE-RELATED DISEASES RIPK1, RIPK2, RIPK3 CES2 3920/4885CES1 1421/4885TRPM8 2983/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.