SCHEMBL30593264

SCHEMBL30593264

NC(=O)N1CCc2cc(-c3ccccc3)ccc2C1c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
CYP11B2 P19099 7/20 0.45
CYP3A4 P08684 1/20 0.45
CYP11B1 P15538 5/20 0.44
CA12 O43570 5/20 0.44
CA1 P00915 5/20 0.44
CA2 P00918 5/20 0.44
CA7 P43166 5/20 0.44
CA9 Q16790 5/20 0.44
CA14 Q9ULX7 5/20 0.44
TRPM8 Q7Z2W7 1/20 0.41
LHCGR P22888 1/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31083687 0.79 CYP11B2 (0.44) CYP11B2CYP11B1
SCHEMBL31070639 0.76 TRPM8 (0.43) CYP11B2TRPM8LHCGR
SCHEMBL31083750 0.76 KDR (0.38) ESR1ESR2CYP11B2CYP11B1CA12
SCHEMBL30593227 0.74 ECE1 (0.44) ESR1ESR2
SCHEMBL30593239 0.74 DRD2 (0.41) ESR1ESR2HTR2ACA12CA1
SCHEMBL25604564 0.74 HHAT (0.57) ESR1ESR2CA12CA1CA2
SCHEMBL31083691 0.73 KIF11 (0.41)
SCHEMBL19378992 0.73 TRPM8 (0.43) CYP3A4TRPM8LHCGR
SCHEMBL30593219 0.72 AURKA (0.43)
SCHEMBL29084871 0.72 HSD11B1 (0.40) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed