SCHEMBL30690645

SCHEMBL30690645

Cn1cc(-c2cc3cc(C#N)cnc3n2COCC[Si](C)(C)C)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 6/20 0.35
CCNA2 P20248 5/20 0.34
CDK2 P24941 5/20 0.34
CCNK O75909 4/20 0.34
CDK12 Q9NYV4 4/20 0.34
SCN2A Q99250 1/20 0.34
CECR2 Q9BXF3 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33
CSNK1G2 P78368 1/20 0.33
EGLN2 Q96KS0 1/20 0.33
SCN9A Q15858 1/20 0.33
DGAT1 O75907 1/20 0.32
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
PIM1 P11309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30690764 0.81 CHEK1 (0.39) DGAT1PIM1
SCHEMBL30690772 0.79 PTGER4 (0.34) IRAK4DGAT1
SCHEMBL30690778 0.79 PTGER4 (0.34) IRAK4DGAT1
SCHEMBL30690669 0.78 IRAK4 (0.31) IRAK4
SCHEMBL30877441 0.78 BAZ2B (0.38) CCNA2CDK2CCNKCDK12SCN2A
SCHEMBL2320459 0.78 DGAT1 (0.39) DGAT1
SCHEMBL30877382 0.77 PTGER4 (0.33) DGAT1
SCHEMBL1356777 0.76 AURKA (0.33) DGAT1
SCHEMBL30877396 0.76 PGR (0.35) CCNA2CDK2CCNKCDK12SCN2A
SCHEMBL1932350 0.75 NTRK1 (0.34) DGAT1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023247593-A1 PYRROLOPYRIDINE CARBOXAMIDES AND THEIR USES AS PDGFR INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2023-12-28 WO disclosed