SCHEMBL30712646

SCHEMBL30712646

COC(=O)c1cc(-c2ccccc2)c(-c2ccccc2)nn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
GABRA1 P14867 2/20 0.55
GABRG2 P18507 2/20 0.55
GABRB3 P28472 2/20 0.55
GABRA3 P34903 2/20 0.55
GABRA5 P31644 1/20 0.55
KDM4E B2RXH2 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
EGFR P00533 1/20 0.46
PTGS1 P23219 1/20 0.46
TP53 P04637 1/20 0.44
THRB P10828 1/20 0.44
MAPT P10636 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
SOAT1 P35610 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26986579 1.00 ALDH1A1 (0.55) ALDH1A1GABRA1GABRG2GABRB3GABRA3
SCHEMBL1752957 0.84 ALDH1A1 (0.55) ALDH1A1GABRA1GABRG2GABRB3GABRA3
SCHEMBL26986682 0.83 ALDH1A1 (0.46) ALDH1A1KDM4ESMN1; SMN2GAAHPGD
SCHEMBL30712643 0.83 ALDH1A1 (0.46) ALDH1A1KDM4ESMN1; SMN2GAAHPGD
SCHEMBL28241571 0.76 GABRA1 (0.50) ALDH1A1GABRA1GABRG2GABRB3GABRA3
SCHEMBL2830890 0.76 ALDH1A1 (0.53) ALDH1A1GABRA1GABRG2GABRB3GABRA3
SCHEMBL5223497 0.75 SMN1; SMN2 (0.54) ALDH1A1KDM4ESMN1; SMN2MAPTGAA
Cyclopropane SCHEMBL11658000 0.75 ALDH1A1 (0.48) ALDH1A1GABRA1GABRG2GABRB3GABRA3
SCHEMBL13188224 0.74 GRM2 (0.55) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL18115629 0.73 GABRG2 (0.58) ALDH1A1GABRA1GABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024009283-A1 AT2 ANTAGONISTS FOR NON-ADDICTIVE PAIN RELIEF UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2024-01-11 WO disclosed