SCHEMBL5223497

SCHEMBL5223497

COc1ccc(-c2cc(C(=O)O)nnc2-c2ccc(OC)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.54
ALDH1A1 P00352 2/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
RECQL P46063 1/20 0.54
CFTR P13569 2/20 0.47
MCL1 Q07820 2/20 0.47
BACE1 P56817 1/20 0.46
KDM4E B2RXH2 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
MAP4K4 O95819 1/20 0.46
GAA P10253 1/20 0.46
ALPL P05186 1/20 0.46
CA9 Q16790 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30712643 0.80 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1HPGDKDM4EL3MBTL1
SCHEMBL26986682 0.80 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1HPGDKDM4EL3MBTL1
SCHEMBL5224281 0.79 PTGS2 (0.57) SMN1; SMN2ALDH1A1MAPTHPGDKDM4E
SCHEMBL5227063 0.78 RAB9A (0.63) SMN1; SMN2ALDH1A1MAPTHPGDKDM4E
SCHEMBL5223978 0.77 GAA (0.50) SMN1; SMN2ALDH1A1MAPTHPGDKDM4E
SCHEMBL5227004 0.76 NPC1 (0.62) SMN1; SMN2ALDH1A1MAPTBACE1KDM4E
SCHEMBL4804463 0.76 KDM1A (0.58) SMN1; SMN2ALDH1A1MAPTHPGDKDM4E
SCHEMBL5222119 0.76 KMT2A (0.44) SMN1; SMN2ALDH1A1MAPTKDM4EL3MBTL1
SCHEMBL5225103 0.75 PTGS2 (0.48) SMN1; SMN2ALDH1A1MAPTHPGDKDM4E
SCHEMBL30712646 0.75 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1MAPTHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1300399-B1 PHENYLPYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME KOWA CO (JP) 2007-08-22 EP disclosed
US-6664256-B1 Interleukin- 1 beta inhibitors KOWA CO., LTD. (JP) 2003-12-16 US disclosed
EP-1300399-A1 PHENYLPYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME Kowa Co., Ltd. (JP) 2003-04-09 EP disclosed