SCHEMBL30714715

SCHEMBL30714715

Cc1ncc(COc2ccc3nn(C)c(C(=O)NC4CCOCC4)c3c2)s1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GABRA5 P31644 3/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
HTR3A P46098 2/20 0.37
METTL3 Q86U44 1/20 0.37
RIPK1 Q13546 1/20 0.36
CNR2 P34972 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SCN9A Q15858 1/20 0.36
AXL P30530 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30714633 0.91 SLC6A5 (0.41) GABRA5HTR3AALDH1A1
SCHEMBL31539881 0.89 HTR3A (0.34) NPC1RAB9AHTR3AALDH1A1
SCHEMBL30714616 0.84 NPC1 (0.40) HPGDSNPC1RAB9AGABRA5HTR3A
SCHEMBL30714661 0.82 MMP3 (0.38) CNR2ALDH1A1SCN9A
SCHEMBL30714672 0.82 RAB9A (0.43) HPGDSNPC1RAB9AGABRA5HTR3A
SCHEMBL26696031 0.81 MCHR1 (0.37) NPC1RAB9AALDH1A1
SCHEMBL26874831 0.81 MCHR1 (0.38) RAB9AALDH1A1
SCHEMBL30714626 0.81 PARG (0.34) NPC1RAB9AGABRA5ALDH1A1
SCHEMBL30714670 0.80 MCHR1 (0.40) NPC1RAB9AALDH1A1
SCHEMBL30714611 0.80 PARG (0.36) NPC1RAB9AALDH1A1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS UNIV LEUVEN KATH (BE) 2025-12-11 US disclosed
EP-4499624-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS Katholieke Universiteit Leuven KU Leuven Research & Development (BE) 2025-02-05 EP disclosed
WO-2023230540-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS TRPV3, TRPM2, TRPV1 HPGDS 671/4885NPC1 349/4885RAB9A 2614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.