SCHEMBL30737249

SCHEMBL30737249

CNC(=O)c1ccc2c(Oc3ccc(C(=O)Cl)cn3)cccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.50
PLK1 P53350 1/20 0.43
PSMD14 O00487 1/20 0.43
STAMBP O95630 1/20 0.43
COPS5 Q92905 1/20 0.43
NCEH1 Q6PIU2 1/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RGS12 O14924 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
KDR P35968 3/20 0.38
AURKA O14965 1/20 0.38
LCK P06239 1/20 0.38
MET P08581 1/20 0.38
TEK Q02763 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30737363 0.90 HPGDS (0.51) HPGDSPLK1PSMD14STAMBPCOPS5
SCHEMBL30737479 0.89 HPGDS (0.53) HPGDSPLK1PSMD14STAMBPCOPS5
SCHEMBL30737390 0.82 PLK1 (0.44) HPGDSPLK1LMNAOPRM1OPRD1
SCHEMBL30737317 0.80 F10 (0.52) MEN1KMT2AMAPTOPRM1OPRD1
SCHEMBL30737175 0.78 SORT1 (0.64) HPGDSOPRM1OPRD1
SCHEMBL23474091 0.75 MAPK1 (0.45) HPGDSPSMD14LMNAMEN1KMT2A
SCHEMBL4257164 0.72 NNMT (0.50) LMNAMEN1KMT2ARGS12MAPT
SCHEMBL30737283 0.71 PLK1 (0.45) HPGDSPLK1LMNAMAPTOPRM1
SCHEMBL30737273 0.70 PLK1 (0.47) HPGDSPLK1LMNAMEN1KMT2A
SCHEMBL19205985 0.70 ALDH1A1 (0.53) HPGDSLMNAMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4543858-A1 BIFUNCTIONAL MOLECULES THAT SELECTIVELY INDUCE DEGRADATION OF EXTRACELLULAR TARGETS IN LYSOSOMES Draupnir Bio ApS (DK) 2025-04-30 EP disclosed
WO-2023247754-A1 BIFUNCTIONAL MOLECULES THAT SELECTIVELY INDUCE DEGRADATION OF EXTRACELLULAR TARGETS IN LYSOSOMES DRAUPNIR BIO APS (DK) 2023-12-28 WO disclosed