SCHEMBL30799557

SCHEMBL30799557

COC(=O)c1sc2cc[n+]([O-])cc2c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
MAPK1 P28482 2/20 0.44
ALDH1A1 P00352 6/20 0.43
HSD17B10 Q99714 5/20 0.43
KDM4E B2RXH2 5/20 0.43
MAPT P10636 5/20 0.43
GLA P06280 3/20 0.43
HPGD P15428 3/20 0.43
GAA P10253 2/20 0.43
KMT2A Q03164 2/20 0.43
ATM Q13315 2/20 0.43
ALOX15 P16050 2/20 0.43
MEN1 O00255 1/20 0.43
CASP1 P29466 1/20 0.37
HTT P42858 1/20 0.37
CASP7 P55210 1/20 0.37
NCOA1 Q15788 1/20 0.37
RCE1 Q9Y256 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
TSHR P16473 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1808035 0.79 LMNA (0.46) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL1805430 0.76 LMNA (0.69) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL16096073 0.72 LMNA (0.48) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL19283497 0.71 LMNA (0.47) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL30799595 0.71 ALDH1A1 (0.58) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL28370458 0.70 LMNA (0.46) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL25208220 0.69 BCKDK (0.49) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL31015986 0.69 RXFP1 (0.51) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL31015992 0.69 BCKDK (0.49) LMNAMAPK1ALDH1A1HSD17B10KDM4E
SCHEMBL25257143 0.69 RXFP1 (0.51) LMNAMAPK1ALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683042-A Fused tetracyclic compound, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2024-03-12 CN disclosed