SCHEMBL30833643

SCHEMBL30833643

NS(=O)(=O)Cc1ccccc1Nc1nc(Cl)ncc1Cl

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 4/20 0.43
CDK7 P50613 10/20 0.41
CDK9 P50750 9/20 0.41
TRPV1 Q8NER1 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 2/20 0.39
MAPK10 P53779 2/20 0.39
BCL6 P41182 1/20 0.39
MET P08581 1/20 0.38
AURKA O14965 1/20 0.38
AURKB Q96GD4 1/20 0.38
INSR P06213 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833659 0.88 AURKA (0.48) ALKCDK7CDK9TRPV1MAPK8
SCHEMBL30833733 0.88 PIN1 (0.36) ALKCDK7CDK9TRPV1AURKA
SCHEMBL30833796 0.88 IGF1R (0.46) ALKCDK7CDK9TRPV1MAPK8
SCHEMBL30833765 0.88 PKMYT1 (0.38) ALKCDK7CDK9TRPV1AURKA
SCHEMBL29904714 0.87 ALK (0.48) ALKCDK7CDK9MAPK8BCL6
SCHEMBL26906809 0.87 ALK (0.48) ALKCDK7CDK9MAPK8BCL6
SCHEMBL27238023 0.85 ALK (0.40) ALKCDK7CDK9MAPK8MAPK9
SCHEMBL30833703 0.84 TRPV1 (0.47) CDK7CDK9TRPV1AURKB
SCHEMBL29904758 0.83 ALK (0.41) ALKMAPK9MAPK10INSR
SCHEMBL2061884 0.82 BPTF (0.44) ALKCDK7CDK9MAPK8MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed