SCHEMBL30833765

SCHEMBL30833765

Cc1cnc(Cl)nc1Nc1ccccc1CS(N)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKMYT1 Q99640 1/20 0.38
CDK7 P50613 1/20 0.37
CDK9 P50750 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
GAA P10253 1/20 0.36
AURKA O14965 2/20 0.35
YTHDC1 Q96MU7 2/20 0.35
ALK Q9UM73 2/20 0.35
INSR P06213 1/20 0.35
S100A9 P06702 1/20 0.34
MAPT P10636 1/20 0.34
AURKB Q96GD4 1/20 0.34
IGF1R P08069 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
LMNA P02545 1/20 0.34
PIN1 Q13526 1/20 0.34
LRRK2 Q5S007 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833643 0.88 ALK (0.43) CDK7CDK9TRPV1AURKAALK
SCHEMBL30833659 0.85 AURKA (0.48) CDK7CDK9TRPV1AURKAALK
SCHEMBL30833796 0.85 IGF1R (0.46) CDK7CDK9TRPV1AURKAALK
SCHEMBL30833733 0.85 PIN1 (0.36) CDK7CDK9TRPV1GAAAURKA
SCHEMBL30833703 0.82 TRPV1 (0.47) CDK7CDK9TRPV1YTHDC1AURKB
SCHEMBL30833754 0.78 MAPT (0.36) CDK9GAAAURKAYTHDC1MAPT
SCHEMBL25005167 0.78 BRD4 (0.43) PKMYT1CDK7CDK9AURKAALK
SCHEMBL29904714 0.78 ALK (0.48) CDK7CDK9YTHDC1ALKINSR
SCHEMBL31147615 0.78 BRD4 (0.43) PKMYT1CDK7CDK9AURKAALK
SCHEMBL26906809 0.78 ALK (0.48) CDK7CDK9YTHDC1ALKINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed