SCHEMBL30833733

SCHEMBL30833733

NS(=O)(=O)Cc1ccccc1Nc1nc(Cl)ncc1I

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 3/20 0.36
TRPV1 Q8NER1 1/20 0.36
S100A9 P06702 1/20 0.34
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
YTHDC1 Q96MU7 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
ALK Q9UM73 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
BPTF Q12830 1/20 0.32
KAT2B Q92831 1/20 0.32
GAA P10253 1/20 0.31
CA12 O43570 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833643 0.88 ALK (0.43) TRPV1AURKAAURKBALKCDK7
SCHEMBL30833796 0.85 IGF1R (0.46) TRPV1AURKAAURKBMEN1KMT2A
SCHEMBL30833765 0.85 PKMYT1 (0.38) PIN1TRPV1S100A9AURKAAURKB
SCHEMBL30833659 0.85 AURKA (0.48) TRPV1AURKAAURKBMAPTTP53
SCHEMBL30833703 0.82 TRPV1 (0.47) TRPV1AURKBYTHDC1CDK7CDK9
SCHEMBL30833645 0.78 PIN1 (0.36) PIN1MAPTYTHDC1MEN1KMT2A
SCHEMBL30833663 0.78 PIN1 (0.36) PIN1MAPTYTHDC1MEN1KMT2A
SCHEMBL22807434 0.76 EGFR (0.42) PIN1MAPTTP53MEN1KMT2A
SCHEMBL30833629 0.76 EGFR (0.42) PIN1MAPTTP53MEN1KMT2A
SCHEMBL29549370 0.76 EGFR (0.42) PIN1MAPTTP53MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed