SCHEMBL3105969

SCHEMBL3105969

Clc1cccc(C(Br)c2ccc(Cc3ccc(CBr)cc3)cc2)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
SLC2A1 P11166 2/20 0.34
PGR P06401 1/20 0.34
PNMT P11086 2/20 0.33
TAAR1 Q96RJ0 2/20 0.33
AOC3 Q16853 1/20 0.33
ACP3 P15309 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
LTA4H P09960 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3107946 0.81 TRPA1 (0.50) ALDH1A1LTA4H
SCHEMBL3110394 0.80 PNMT (0.37) SLC2A1PNMTTAAR1AOC3ACP3
SCHEMBL17061793 0.79 ACP3 (0.46) PNMTAOC3ACP3IDO1TDO2
SCHEMBL7521832 0.77 ACP3 (0.50) ADRB1ADRB3ACP3IDO1TDO2
SCHEMBL3105616 0.74 SLC6A2 (0.37) TAAR1IDO1ALDH1A1
SCHEMBL3113885 0.73 KEAP1 (0.38) TAAR1IDO1ALDH1A1LTA4H
SCHEMBL3105632 0.73 IDO1 (0.36) TAAR1IDO1TDO2ALDH1A1
SCHEMBL3103812 0.72 SLC6A2 (0.37) ALDH1A1
SCHEMBL13496520 0.72 CALM1 (0.55) ALDH1A1LTA4H
SCHEMBL3107011 0.71 TSHR (0.42) PNMTTAAR1AOC3ACP3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2163553-B1 ARENE CONNECTED POLYAMINE MACRORING DERIVATIVES, PREPARATION METHODS AND PHARMACEUTICAL USES THEREOF BEIJING MOLECULE SCIENCE AND TECHNOLOGY CO LTD (CN) 2013-12-25 EP disclosed
EP-2163553-A1 ARENE CONNECTED POLYAMINE MACRORING DERIVATIVES, PREPARATION METHODS AND PHARMACEUTICAL USES THEREOF Beijing Molecule Science and Technology Co., Ltd. (CN) 2010-03-17 EP disclosed