Methylamine

Methylamine

SCHEMBL313813

CN.N.O

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Methylamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylamine SCHEMBL4335369 1.00
Methylamine SCHEMBL5492498 0.89
Methylamine SCHEMBL3240364 0.89
Methylamine SCHEMBL8507247 0.89
Methylamine SCHEMBL8644698 0.89
Methylamine SCHEMBL6130807 0.89
Methylamine SCHEMBL9853401 0.89
Methylamine SCHEMBL8931568 0.89
Methylamine SCHEMBL538799 0.89
Methylamine SCHEMBL2341548 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 177 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12031132-B2 Systems and methods for the treatment of hemoglobinopathies EDITAS MEDICINE, INC. (US) 2024-07-09 US disclosed
EP-4392076-A1 SIRP-ALPHA ANTIBODIES AND CONJUGATES Tallac Therapeutics, Inc. (US) 2024-07-03 EP disclosed
EP-4388103-A1 NECTIN-4 ANTIBODIES AND CONJUGATES Tallac Therapeutics, Inc. (US) 2024-06-26 EP disclosed
CN-118215485-A Branched trisaccharide modified nucleic acid compounds 诺华股份有限公司 2024-06-18 CN disclosed
CN-118215484-A Staggered trisaccharide modified nucleic acid compounds 诺华股份有限公司 2024-06-18 CN disclosed
US-20240191197-A1 MODIFIED CELLS AND METHODS FOR THE TREATMENT OF HEMOGLOBINOPATHIES EDITAS MEDICINE, INC. (US) 2024-06-13 US disclosed
US-20240191242-A1 TRANSGLUTAMINASE-MEDIATED CONJUGATION HORIZON TECHNOLOGY FINANCE CORPORATION 2024-06-13 US disclosed
WO-2024105654-A1 METHODS AND COMPOSITIONS INCLUDING CONJUGATED DNAZYMES 1E THERAPEUTICS, LTD. (IL) 2024-05-23 WO disclosed
EP-3583211-B1 METHOD FOR THE SYNTHESIS OF DNA CONJUGATES BY MICELLAR CATALYSIS UNIV DORTMUND TECH (DE) 2024-04-10 EP disclosed
US-11920136-B2 Transglutaminase-mediated conjugation Tallac Therapeutics, Inc. (US) 2024-03-05 US disclosed
WO-2000071559-A9 METHOD FOR DEBLOCKING OF LABELED OLIGONUCLEOTIDES INVITROGEN CORP (US) 2001-06-21 WO disclosed
EP-1091972-A1 REUSABLE SOLID SUPPORT FOR OLIGONUCLEOTIDE SYNTHESIS UNIVERSITY TECHNOLOGIES INTERNATIONAL INC. (CA) 2001-04-18 EP disclosed
WO-2000071559-A1 METHOD FOR DEBLOCKING OF LABELED OLIGONUCLEOTIDES INVITROGEN CORPORATION (US) 2000-11-30 WO disclosed
US-6043353-A FOR SOLID PHASE SYNTHESIS UNIVERSITY TECHNOLOGIES INTERNATIONAL, INC. (CA) 2000-03-28 US disclosed
WO-2000001711-A1 REUSABLE SOLID SUPPORT FOR OLIGONUCLEOTIDE SYNTHESIS UNIVERSITY TECHNOLOGIES INTERNATIONAL INC. (CA) 2000-01-13 WO disclosed
EP-0876390-A1 REUSABLE SOLID SUPPORT FOR OLIGONUCLEOTIDE SYNTHESIS, PROCESS FOR PRODUCTION THEREOF AND PROCESS FOR USE THEREOF UNIVERSITY TECHNOLOGIES INTERNATIONAL INC. (CA) 1998-11-11 EP disclosed
EP-0866072-A1 Processes for purifying synthetic oligonucleotides Beckman Coulter, Inc. (US) 1998-09-23 EP disclosed
US-5770723-A HIGH SPEED DEPROTECTION AND CLEAVAGE WITH METHYLAMINE; ADDINGSODIUM CHLORIDE AND/OR AMMONIUM ACETATE BECKMAN INSTRUMENTS, INC. 1998-06-23 US disclosed
WO-1997023496-A1 REUSABLE SOLID SUPPORT FOR OLIGONUCLEOTIDE SYNTHESIS, PROCESS FOR PRODUCTION THEREOF AND PROCESS FOR USE THEREOF UNIVERSITY TECHNOLOGIES INTERNATIONAL INC. (CA) 1997-07-03 WO disclosed
US-5601979-A SOLID PHASE DNA SYNTHESIS CPG, INC. (US) 1997-02-11 US disclosed