Benzylimidazole

Benzylimidazole

SCHEMBL3139033

O=C(O)C(F)(F)F.c1ccc(Cn2ccnc2)cc1

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 8/20 0.73
CYP11B1 P15538 6/20 0.73
CYP19A1 P11511 5/20 0.73
CYP11B2 P19099 5/20 0.73
CYP1A2 P05177 3/20 0.73
CYP3A4 P08684 2/20 0.73
CYP2D6 P10635 2/20 0.73
POLB P06746 1/20 0.73
MAPT P10636 1/20 0.73
QPCT Q16769 1/20 0.73
CYP4Z1 Q86W10 1/20 0.73
QPCTL Q9NXS2 1/20 0.73
CYP17A1 P05093 1/20 0.60
USP2 O75604 1/20 0.55
LMNA P02545 1/20 0.55
MEN1 O00255 1/20 0.55
CYP2C19 P33261 1/20 0.55
KMT2A Q03164 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzylimidazole SCHEMBL16236718 0.86 TBXAS1 (0.80) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL16700262 0.85 CYP11B1 (0.69) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL414 0.85 CYP11B1 (1.00) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
SCHEMBL22063900 0.85 CYP11B1 (1.00) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Trifluoroacetic Acid SCHEMBL8307090 0.84 CYP11B1 (0.74) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL411827 0.84 CYP11B1 (0.96) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL16237308 0.84 CYP11B1 (0.96) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL29239318 0.84 CYP11B1 (0.96) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL31453527 0.84 CYP11B1 (0.96) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2
Benzylimidazole SCHEMBL3786782 0.84 CYP11B1 (0.96) TBXAS1CYP11B1CYP19A1CYP11B2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3244987-B1 SEPARATIONS WITH IONIC LIQUID SOLVENTS CHEVRON PHILLIPS CHEMICAL CO LP (US) 2022-06-22 EP claimed
EP-3244987-A1 SEPARATIONS WITH IONIC LIQUID SOLVENTS Chevron Phillips Chemical Company LP (US) 2017-11-22 EP claimed
US-20150133711-A1 Separations With Ionic Liquid Solvents CHEVRON PHILLIPS CHEMICAL COMPANY LP 2015-05-14 US claimed
EP-3244987-B1 SEPARATIONS WITH IONIC LIQUID SOLVENTS CHEVRON PHILLIPS CHEMICAL CO LP (US) 2022-06-22 EP disclosed
US-10227274-B2 Separations with ionic liquid solvents CHEVRON PHILLIPS CHEMICAL COMPANY LP (US) 2019-03-12 US disclosed
EP-3244987-A1 SEPARATIONS WITH IONIC LIQUID SOLVENTS Chevron Phillips Chemical Company LP (US) 2017-11-22 EP disclosed
US-20150133711-A1 Separations With Ionic Liquid Solvents CHEVRON PHILLIPS CHEMICAL COMPANY LP 2015-05-14 US disclosed
EP-1858909-B1 SYNTHESIS OF OLIGONUCLEOTIDES GIRINDUS AG (DE) 2014-09-10 EP disclosed
EP-1828218-B1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR GIRINDUS AG (DE) 2014-04-30 EP disclosed
US-20130281682-A1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR GIRINDUS AG (DE) 2013-10-24 US disclosed
US-20120322994-A1 SYNTHESIS OF OLIGONUCLEOTIDES GIRINDUS AG (DE) 2012-12-20 US disclosed
US-20120316328-A1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR GIRINDUS AG (DE) 2012-12-13 US disclosed
US-20110065909-A1 SYNTHESIS OF OLIGONUCLEOTIDES GIRINDUS AG (DE) 2011-03-17 US disclosed
US-20100081802-A1 Synthesis of Phosphitylated Compounds Using a Quaternary Heterocyclic Activator GIRINDUS AG (DE) 2010-04-01 US disclosed
EP-1828218-A1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR Girindus AG (DE) 2007-09-05 EP disclosed
WO-2006064039-A1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR GIRINDUS AG (DE) 2006-06-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110065909-A1 SYNTHESIS OF OLIGONUCLEOTIDES RNGTT, CPSF1, CPSF6 TBXAS1 454/4885CYP11B1 2759/4885CYP19A1 768/4885
US-20100081802-A1 Synthesis of Phosphitylated Compounds Using a Quaternary Heterocyclic Activator ARAF, ATIC, PFKFB3 TBXAS1 2582/4885CYP11B1 3876/4885CYP19A1 2889/4885
US-20120316328-A1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR ARAF, ATIC, PFKFB3 TBXAS1 2817/4885CYP11B1 4127/4885CYP19A1 3224/4885
US-20120322994-A1 SYNTHESIS OF OLIGONUCLEOTIDES RNGTT, CPSF1, CPSF6 TBXAS1 454/4885CYP11B1 2759/4885CYP19A1 768/4885
US-20130281682-A1 SYNTHESIS OF PHOSPHITYLATED COMPOUNDS USING A QUATERNARY HETEROCYCLIC ACTIVATOR ARAF, ATIC, HK2 TBXAS1 2516/4885CYP11B1 4175/4885CYP19A1 3442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.