SCHEMBL3141113

SCHEMBL3141113

O=C(O)Oc1cc2cnccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.51
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
HRH4 Q9H3N8 1/20 0.44
CNR2 P34972 1/20 0.41
NAMPT P43490 11/20 0.41
CYP2C9 P11712 3/20 0.38
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
MAPT P10636 1/20 0.37
SNCA P37840 1/20 0.37
MAP2K1 Q02750 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4038601 0.87 DAO (0.51) DAOPDE3BPDE3AHRH4HDAC3
SCHEMBL28761709 0.86 DAO (0.50) DAOPDE3BPDE3AHRH4CNR2
SCHEMBL4033217 0.86 DAO (0.50) DAOPDE3BPDE3AHRH4CNR2
SCHEMBL1833251 0.76 KDM4E (0.55) DAOMAPT
SCHEMBL29079873 0.75 DAO (0.49) DAOPDE3BPDE3AHRH4CNR2
SCHEMBL168527 0.75 DAO (0.58) DAOPDE3BPDE3AHRH4CNR2
SCHEMBL5155719 0.73 SMAD3 (0.57) HRH4
SCHEMBL1824754 0.73 HCAR2 (0.32)
SCHEMBL4036292 0.73 DAO (0.50) DAOHRH4HDAC3HDAC1HDAC2
SCHEMBL3381954 0.72 FLT3 (0.48) HRH4HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2820017-B1 PYRIDINYL AND PYRIMIDINYL SULFOXIDE AND SULFONE DERIVATIVES GENENTECH INC (US) 2016-12-21 EP claimed
EP-1636224-B1 PYRROLOPYRIDINE-2-CARBOXYLIC ACID AMIDE INHIBITORS OF GLYCOGEN PHOSHORYLASE PROSIDION LTD (GB) 2010-07-14 EP claimed
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed