SCHEMBL3150987

SCHEMBL3150987

CNC1(COc2cncc(-c3ccc(-c4nn[nH]n4)cc3)c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
XDH P47989 4/20 0.46
AKT1 P31749 1/20 0.46
TP53 P04637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP19A1 P11511 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ADH5 P11766 1/20 0.41
SLC22A12 Q96S37 1/20 0.40
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3772959 0.99 XDH (0.45) XDHAKT1TP53ALDH1A1CYP19A1
SCHEMBL3150879 0.91 SLC22A12 (0.47) XDHAKT1ALDH1A1SLC22A12
Hydrochloric Acid SCHEMBL3778977 0.90 SLC22A12 (0.47) XDHAKT1ALDH1A1SLC22A12
SCHEMBL3141790 0.81 CHRNB2 (0.48) XDH
Hydrochloric Acid SCHEMBL3768153 0.81 ALDH1A1 (0.41) XDHTP53ALDH1A1CYP19A1CYP2C9
Hydrochloric Acid SCHEMBL3773084 0.80 CHRNB2 (0.47) XDH
SCHEMBL3145280 0.80 CHRNB1 (0.49) AKT1
SCHEMBL3150922 0.80 CHRNB1 (0.49) AKT1
SCHEMBL3151157 0.80 CHRNB1 (0.49) CYP2C9
SCHEMBL3147229 0.80 CHRNB2 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed