SCHEMBL3150879

SCHEMBL3150879

CNC1(COc2cncc(-c3cccc(-c4nn[nH]n4)c3)c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.47
GP6 Q9HCN6 2/20 0.44
XDH P47989 1/20 0.44
EGLN1 Q9GZT9 2/20 0.43
CYSLTR2 Q9NS75 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
ALDH1A1 P00352 1/20 0.40
AKT1 P31749 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
CYP2A6 P11509 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3778977 0.99 SLC22A12 (0.47) SLC22A12GP6XDHEGLN1CYSLTR2
SCHEMBL3150987 0.91 XDH (0.46) SLC22A12XDHALDH1A1AKT1
Hydrochloric Acid SCHEMBL3772959 0.90 XDH (0.45) SLC22A12XDHALDH1A1AKT1
Hydrochloric Acid SCHEMBL3774374 0.82 IDO1 (0.40) SLC22A12GP6XDHEGLN1ALDH1A1
SCHEMBL3150645 0.80 CYP11B1 (0.47)
SCHEMBL3142735 0.80 S1PR1 (0.38) SLC22A12XDH
SCHEMBL3147229 0.80 CHRNB2 (0.49)
SCHEMBL3147306 0.79 INPPL1 (0.43) SLC22A12XDHAKT1
SCHEMBL3137054 0.79 CYP11B2 (0.39) AKT1
SCHEMBL3146014 0.79 CHRNB1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed