SCHEMBL3175406

SCHEMBL3175406

CCC(CCC(N)=O)SC(C)=O

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
KMT2A Q03164 1/20 0.42
DPP4 P27487 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2404276 0.78
SCHEMBL6398895 0.73 EPHX1 (0.45) KMT2A
SCHEMBL4364680 0.71 ENPEP (0.37) KMT2A
SCHEMBL14930200 0.70 ALDH1A1 (0.40)
SCHEMBL3716659 0.69 KMT2A (0.46) ALOX15BLMPMP22KMT2ADPP4
SCHEMBL8722957 0.68 CA2 (0.43) ALOX15BLMPMP22KMT2ADPP4
SCHEMBL10837425 0.68 CA2 (0.39) CA1CA2
SCHEMBL6079159 0.68 NOS3 (0.30)
SCHEMBL1747943 0.67
SCHEMBL7770036 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660507-B9 PROTEASOME INHIBITORS AND METHODS OF USING THE SAME CEPHALON INC (US) 2010-03-24 EP claimed
EP-1660507-B1 PROTEASOME INHIBITORS AND METHODS OF USING THE SAME CEPHALON INC (US) 2009-08-05 EP claimed