SCHEMBL3227728

SCHEMBL3227728

Nc1cc(NCc2c(F)cccc2F)nc2c1nc(C(F)(F)F)c(=O)n2C1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 6/20 0.37
SCN1A P35498 3/20 0.37
SCN5A Q14524 2/20 0.37
CD38 P28907 3/20 0.34
CYP3A4 P08684 2/20 0.34
KCNH2 Q12809 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
STIM1 Q13586 1/20 0.34
ORAI1 Q96D31 1/20 0.34
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
PDE2A O00408 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7944093 0.81 STIM1 (0.38) CD38CYP3A4KCNH2STIM1ORAI1
SCHEMBL7945084 0.79 CYP1A2 (0.47) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL3227997 0.74 CYP11B2 (0.37) CYP3A4KCNH2CYP1A2CYP2D6CYP2C9
SCHEMBL7943760 0.70 CD38 (0.37) CD38CYP3A4CYP1A2CYP2C19STIM1
SCHEMBL7937855 0.69 CYP1A2 (0.37) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7937858 0.69 CYP1A2 (0.49) CYP3A4CYP1A2CYP2D6CYP2C9MEN1
SCHEMBL7937752 0.64 ADORA2A (0.39) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7945503 0.64 TLR9 (0.37) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL7937861 0.61 TLR9 (0.35) CYP2D6CYP2C19PDE4APDE4BPDE4C
SCHEMBL7947006 0.61 ALDH1A1 (0.34) CYP3A4CYP1A2CYP2D6CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed