SCHEMBL7937752

SCHEMBL7937752

CCCn1c(=O)c(-c2nccs2)nc2c(N)cc(NCc3c(F)cccc3F)nc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.39
ADORA1 P30542 4/20 0.39
ADORA2B P29275 3/20 0.39
ADORA3 P0DMS8 2/20 0.35
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
USP2 O75604 5/20 0.32
CYP1A2 P05177 5/20 0.32
CYP3A4 P08684 5/20 0.32
CASP1 P29466 5/20 0.32
CASP7 P55210 5/20 0.32
HSD17B10 Q99714 5/20 0.32
ALDH1A1 P00352 5/20 0.32
HIF1A Q16665 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7937864 0.93 ADORA2A (0.38) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL7943995 0.86 HSF1 (0.36) ADORA2AADORA1ADORA3USP2CYP1A2
SCHEMBL7937747 0.85 HSF1 (0.35) ADORA2AADORA1ADORA3USP2CYP1A2
SCHEMBL7944574 0.83 HSF1 (0.36) ADORA2AADORA1ADORA2BADORA3HPGD
SCHEMBL7943760 0.82 CD38 (0.37) ADORA2AADORA1ADORA2BCCNT1CDK9
SCHEMBL7944093 0.80 STIM1 (0.38) ADORA2AADORA1ADORA2BCCNT1CDK9
SCHEMBL7944078 0.76 PDE4B (0.42) ADORA2AADORA1ADORA2BADORA3PDE4B
SCHEMBL7944114 0.70 PDE4B (0.48) ADORA2AADORA1ADORA2BADORA3PDE4A
SCHEMBL7946794 0.69 ADORA1 (0.39) ADORA2AADORA1ADORA2BADORA3PDE4B
SCHEMBL7945987 0.69 TYRO3 (0.36) USP2CYP1A2CASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed