SCHEMBL3229178

SCHEMBL3229178

Cc1cc2ccccc2n1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.43
TP53 P04637 3/20 0.40
KDM4E B2RXH2 3/20 0.40
KMT2A Q03164 7/20 0.39
TSHR P16473 2/20 0.38
NOS2 P35228 1/20 0.38
MEN1 O00255 6/20 0.37
MAPT P10636 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
NPC1 O15118 1/20 0.37
HSP90AA1 P07900 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16507810 0.76 CYP1A2 (0.44) TP53KDM4EMAPTCYP1A2CYP3A4
SCHEMBL14159651 0.75 DAO (0.44) TP53KDM4EKMT2AALDH1A1PKM
SCHEMBL154592 0.74 KMT2A (0.55) SLC6A2TP53KDM4EKMT2AMEN1
SCHEMBL29378766 0.74 KMT2A (0.55) SLC6A2TP53KDM4EKMT2AMEN1
SCHEMBL7678437 0.74 SLC6A2 (0.44) SLC6A2TP53KDM4EKMT2ATSHR
SCHEMBL8598225 0.74 NOS2 (0.43) TP53KDM4EKMT2ATSHRNOS2
SCHEMBL3008864 0.73 DAO (0.52) SLC6A2TP53KDM4EKMT2ATSHR
SCHEMBL3973543 0.73 SLC6A2 (0.43) SLC6A2TP53KDM4EKMT2ATSHR
SCHEMBL18525155 0.73 SLC6A2 (0.43) SLC6A2TP53KDM4EKMT2ATSHR
SCHEMBL6114342 0.73 SLC6A2 (0.43) SLC6A2TP53KDM4EKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2142516-B1 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS SANOFI SA (FR) 2012-12-26 EP claimed
US-8258130-B2 Pyrimidine hydrazide compounds as PGDS inhibitors SANOFI (FR) 2012-09-04 US claimed
US-20100048568-A1 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS SANOFI-AVENTIS (FR) 2010-02-25 US claimed
EP-2142516-A1 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS Sanofi-Aventis (FR) 2010-01-13 EP claimed
WO-2008121670-A1 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS SANOFI-AVENTIS (FR) 2008-10-09 WO claimed
WO-2025056724-A1 IMINOAMIDE-TYPE COMPOUNDS AS LIGANDS FOR COPPER-CATALYZED COUPLING REACTIONS OF (HETERO)ARYL HALIDES BAYER AKTIENGESELLSCHAFT (DE) 2025-03-20 WO disclosed
WO-2025056725-A1 PROCESS FOR THE PREPARATION OF HALOGENATED PHENOLS VIA COPPER-CATALYZED COUPLING REACTIONS OF HALOGENATED ARYL-HALIDES BAYER AKTIENGESELLSCHAFT (DE) 2025-03-20 WO disclosed
US-20230276696-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORP (US) 2023-08-31 US disclosed
US-11716898-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2023-08-01 US disclosed
US-11678565-B2 Organic electroluminescent materials and devices UNIVERSAL DISPLAY CORPORATION (US) 2023-06-13 US disclosed
US-11114626-B2 Metal compounds, methods, and uses thereof ARIZONA BOARD OF REGENTS ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2021-09-07 US disclosed
US-20200295276-A1 Organic Electroluminescent Materials and Devices UNIVERSAL DISPLAY CORP (US) 2020-09-17 US disclosed
WO-1997004777-A1 USE OFF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-02-13 WO disclosed
WO-1996026183-A1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS NOVARTIS AG (CH) 1996-08-29 WO disclosed
EP-0635269-A1 Use of N-(Pyridinyl)-1H-Indol-1-Amines for the preparation of a medicament for the treatment of obsessive-compulsive disorders HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1995-01-25 EP disclosed
US-5356910-A Use of N-(pyridinyl)-1H-indol-1-amines for the treatment of obsessive-compulsive disorder HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-10-18 US disclosed
US-5039811-A Analgesics, antidepressants, memory activators; condensation, reduction HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-13 US disclosed
EP-0397040-A2 N-heteroaryl-4-quinolinamines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1990-11-14 EP disclosed
US-4970218-A ANALGESIC, ANTIDEPRESSANT, MEMORY ENHANCEMENT HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-11-13 US disclosed
US-4916135-A ANALGESICS, ALZHEIMER*S HOECHST ROUSSEL PHARMACEUTICALS INC. (US) 1990-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11716898-B2 Organic electroluminescent materials and devices OCIAD2, OCIAD1, JUND SLC6A2 1328/4885TP53 3742/4885KDM4E 2637/4885
US-11678565-B2 Organic electroluminescent materials and devices OCIAD1, OCIAD2, OPRD1 SLC6A2 3013/4885TP53 3538/4885KDM4E 3475/4885
US-11114626-B2 Metal compounds, methods, and uses thereof SOD1, SOD3, AOX1 SLC6A2 1678/4885TP53 3013/4885KDM4E 4380/4885
US-20100048568-A1 PYRIMIDINE HYDRAZIDE COMPOUNDS AS PGDS INHIBITORS HRH2, HRH1, HRH4 SLC6A2 4643/4885TP53 1426/4885KDM4E 2494/4885
US-20200295276-A1 Organic Electroluminescent Materials and Devices OCIAD2, OCIAD1, JUND SLC6A2 1328/4885TP53 3742/4885KDM4E 2637/4885
US-20230276696-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES OCIAD2, OCIAD1, PORCN SLC6A2 2379/4885TP53 3915/4885KDM4E 3190/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.