SCHEMBL3244499

SCHEMBL3244499

CC(C)(C)OC(=O)NCc1cccc(CNC(C(=O)O)C2CCCCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLS O94925 5/20 0.46
ROCK2 O75116 1/20 0.43
BRD4 O60885 2/20 0.42
CREBBP Q92793 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGB1 P05556 1/20 0.42
ITGAV P06756 1/20 0.42
ITGA5 P08648 1/20 0.42
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
EPHX1 P07099 2/20 0.40
F2 P00734 1/20 0.40
CACNA1B Q00975 1/20 0.40
MMP13 P45452 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
HPGD P15428 1/20 0.39
JAK2 O60674 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3457367 0.91 ITGB3 (0.50) ROCK2ITGB3ITGB1ITGAVITGA5
SCHEMBL7947169 0.89 EPHX2 (0.43) GLSROCK2BRD4CREBBPITGB3
SCHEMBL7946795 0.79 GLS (0.48) GLSROCK2BRD4CREBBPCA12
SCHEMBL8202738 0.79 CACNA1B (0.48) ROCK2ITGB3ITGB1ITGAVITGA5
SCHEMBL29228688 0.77 ITGB3 (0.55) ITGB3ITGB1ITGAVITGA5KMT2A
SCHEMBL1410181 0.77 ITGB3 (0.55) ITGB3ITGB1ITGAVITGA5KMT2A
SCHEMBL24732888 0.77 ROCK2 (0.54) GLSROCK2BRD4CREBBPKMT2A
SCHEMBL30779221 0.77 ROCK2 (0.54) GLSROCK2BRD4CREBBPKMT2A
SCHEMBL25048390 0.76 BRD4 (0.47) GLSROCK2BRD4CREBBPKMT2A
SCHEMBL17147653 0.76 ITGB3 (0.53) ITGB3ITGB1ITGAVITGA5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010035032-A1 CALCIUM ION CHANNEL MODULATORS & USES THEREOF LECTUS THERAPEUTICS LIMITED (GB) 2010-04-01 WO disclosed