SCHEMBL3247793

SCHEMBL3247793

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3cc(OC)c(OC)cc3c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.46
GABRA5 P31644 5/20 0.46
GABRA3 P34903 5/20 0.46
GABRA2 P47869 4/20 0.46
GABRA6 Q16445 4/20 0.46
KDM4E B2RXH2 5/20 0.46
ALDH1A1 P00352 4/20 0.46
HPGD P15428 2/20 0.46
GAA P10253 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GABRG2 P18507 3/20 0.44
GABRB3 P28472 3/20 0.44
RET P07949 1/20 0.43
USP2 O75604 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
TUBB4A P04350 2/20 0.40
TUBB P07437 2/20 0.40
TUBA3C P0DPH7 2/20 0.40
TUBA1B P68363 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3248781 0.91 KDM4E (0.40) GABRA1GABRA5GABRA3GABRA2GABRA6
SCHEMBL3250416 0.86 CDK4 (0.46) KDM4EALDH1A1HPGDGAANPSR1
SCHEMBL3254551 0.83 ALDH1A1 (0.52) GABRA1GABRA5GABRA3GABRA2GABRA6
SCHEMBL3249865 0.82 KDM4E (0.40) GABRA1GABRA5GABRA3GABRA2GABRA6
SCHEMBL3248921 0.82 ALDH1A1 (0.41) GABRA1KDM4EALDH1A1HPGDHTT
SCHEMBL3245727 0.82 GABRA1 (0.50) GABRA1GABRA3ALDH1A1HPGDNPSR1
SCHEMBL3251609 0.82 PARP1 (0.44) ALDH1A1HPGDSMN1; SMN2L3MBTL1HSD17B10
SCHEMBL3254034 0.82 ALOX15 (0.47)
SCHEMBL3252529 0.82 ALDH1A1 (0.47) GABRA1GABRA3KDM4EALDH1A1HPGD
SCHEMBL3255332 0.82 ADORA3 (0.40) GABRA1GABRA3KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed