SCHEMBL3255332

SCHEMBL3255332

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(N)cc3c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.40
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
TP53 P04637 2/20 0.40
NPC1 O15118 2/20 0.40
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PARP1 P09874 2/20 0.38
HPGD P15428 4/20 0.37
HSD17B10 Q99714 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GABRA1 P14867 2/20 0.36
GABRB2 P47870 2/20 0.36
NGFR P08138 1/20 0.36
GABRB1 P18505 1/20 0.35
GABRA3 P34903 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253850 0.92 SCN9A (0.38) ADORA3ALDH1A1KDM4ETP53NPC1
SCHEMBL3249476 0.89 ICMT (0.37) ADORA3ALDH1A1KDM4ETP53NPC1
SCHEMBL3245727 0.87 GABRA1 (0.50) ALDH1A1TP53NPC1MAPTRAB9A
SCHEMBL3248921 0.87 ALDH1A1 (0.41) ALDH1A1KDM4ETP53MAPTSMN1; SMN2
SCHEMBL3252529 0.87 ALDH1A1 (0.47) ALDH1A1KDM4ETP53NPC1GAA
SCHEMBL3250516 0.87 TUBB4A (0.36) ADORA3ALDH1A1KDM4ETP53NPC1
SCHEMBL3250557 0.85 MAPT (0.41) ALDH1A1KDM4ETP53MAPTHPGD
SCHEMBL3250586 0.85 HSD17B10 (0.37) ALDH1A1KDM4ETP53GAARAB9A
SCHEMBL3243057 0.85 CHEK1 (0.37) ADORA3ALDH1A1KDM4ETP53HPGD
SCHEMBL3250430 0.84 HSD17B10 (0.45) ALDH1A1KDM4ETP53NPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed