SCHEMBL3250416

SCHEMBL3250416

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3cc(OC)ccc3c12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 5/20 0.46
CCND1 P24385 5/20 0.46
BCHE P06276 2/20 0.45
ACHE P22303 2/20 0.45
ALDH1A1 P00352 5/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 1/20 0.43
CCNE2 O96020 2/20 0.42
CCNE1 P24864 2/20 0.42
CDK2 P24941 2/20 0.42
ROCK2 O75116 1/20 0.42
CAMK2B Q13554 1/20 0.42
CAMK2G Q13555 1/20 0.42
CAMK2D Q13557 1/20 0.42
CAMK2A Q9UQM7 1/20 0.42
KDM4E B2RXH2 6/20 0.41
HPGD P15428 4/20 0.41
HTT P42858 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251609 0.86 PARP1 (0.44) CDK4CCND1ALDH1A1KMT2AMEN1
SCHEMBL3254034 0.86 ALOX15 (0.47) ALOX15
SCHEMBL3249865 0.86 KDM4E (0.40) ALDH1A1KMT2AMEN1HSD17B10KDM4E
SCHEMBL3247793 0.86 GABRA1 (0.46) ALDH1A1HSD17B10KDM4EHPGDHTT
SCHEMBL3254865 0.83 ALDH1A1 (0.47) CDK4CCND1BCHEACHEALDH1A1
SCHEMBL3248781 0.82 KDM4E (0.40) ALDH1A1KMT2AMEN1HSD17B10KDM4E
SCHEMBL3245727 0.80 GABRA1 (0.50) CDK4CCND1ALDH1A1KMT2AMEN1
SCHEMBL3248921 0.80 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1HSD17B10KDM4E
SCHEMBL3252529 0.80 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1HSD17B10ALOX15
SCHEMBL3255332 0.80 ADORA3 (0.40) ALDH1A1KMT2AMEN1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed