SCHEMBL3262268

SCHEMBL3262268

O=C(O)C1(c2ccccc2)C=CC=CC1C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.32
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
CES1 P23141 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4225392 0.84 HTT (0.40) HTTCES1SMN1; SMN2OPRM1OPRD1
SCHEMBL8469874 0.77 AKR1C1 (0.35) AKR1C1LMNAHTTSMN1; SMN2
Hydrochloric Acid SCHEMBL28568646 0.76 HSD11B1 (0.35) AKR1C1LMNAHTT
SCHEMBL9142790 0.76 HSD11B1 (0.35) AKR1C1LMNAHTT
SCHEMBL17707789 0.74 AKR1C1 (0.33) AKR1C1LMNAHTT
SCHEMBL27621152 0.73 LMNA (0.33) AKR1C1LMNAHTTSMN1; SMN2
SCHEMBL20378032 0.68 ALDH1A1 (0.33) LMNAHTTSMN1; SMN2OPRM1
SCHEMBL2274804 0.67 NPC1 (0.41) LMNASMN1; SMN2
SCHEMBL8930987 0.66 CA2 (0.32)
SCHEMBL2276486 0.65 RORC (0.33) HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020548-A1 GLYT1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-02-25 WO disclosed