SCHEMBL3263348

SCHEMBL3263348

Cn1c(=O)c2c(C(C(N)=O)c3nccs3)cccc2n(C)c1=O

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 15/20 0.36
TRPV4 Q9HBA0 4/20 0.35
CTSA P10619 2/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
TRPV3 Q8NET8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3266992 0.87 CNR2 (0.35) TRPA1NPC1PKM
SCHEMBL3266719 0.82 KMT2A (0.35) CTSA
SCHEMBL3264313 0.80 TRPA1 (0.36) TRPA1TRPV4NPC1PKMTRPV3
SCHEMBL9960985 0.80 NPC1 (0.36) NPC1PKM
SCHEMBL3264317 0.74 FFAR2 (0.47) TRPA1NPC1PKM
SCHEMBL4562114 0.73 PORCN (0.44) CTSA
SCHEMBL9960578 0.73 TRPA1 (0.34) TRPA1TRPV4NPC1PKMTRPV3
SCHEMBL667099 0.73 CTSA (0.46) CTSANPC1PKM
SCHEMBL2486908 0.72 TRPA1 (0.33) TRPA1TRPV4NPC1PKM
SCHEMBL662588 0.72 CTSA (0.40) CTSANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010004390-A1 QUINAZOLINE DIONE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS, S.A. (CH) 2010-01-14 WO claimed
WO-2010004390-A1 QUINAZOLINE DIONE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS, S.A. (CH) 2010-01-14 WO disclosed