SCHEMBL2486908

SCHEMBL2486908

Cn1c(=O)c2c(C(C(N)=O)c3nccs3)c(Cl)oc2n(C)c1=O

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 7/20 0.33
TRPV4 Q9HBA0 4/20 0.33
NPC1 O15118 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9960578 0.88 TRPA1 (0.34) TRPA1TRPV4NPC1PKM
SCHEMBL9960985 0.74 NPC1 (0.36) NPC1PKM
SCHEMBL3263348 0.72 TRPA1 (0.36) TRPA1TRPV4NPC1PKM
SCHEMBL2516435 0.66 CTSA (0.30)
SCHEMBL2473502 0.65 PORCN (0.34) TRPA1
SCHEMBL12322879 0.63 TRPA1 (0.43) TRPA1TRPV4
SCHEMBL2475791 0.62 PORCN (0.32) TRPA1PKM
SCHEMBL5585939 0.61 ALDH1A1 (0.43) NPC1
SCHEMBL4562114 0.61 PORCN (0.44)
SCHEMBL665545 0.60 ALOX5 (0.47) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO claimed
WO-2011114184-A1 AMIDES OF HETEROCYCLIC COMPOUNDS AS TRPA1 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-09-22 WO disclosed