SCHEMBL3264313

SCHEMBL3264313

Cn1c(=O)c2c(C(Cc3nccs3)C(N)=O)cccc2n(C)c1=O

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 18/20 0.36
TRPV4 Q9HBA0 4/20 0.35
TRPV3 Q8NET8 1/20 0.33
NPC1 O15118 1/20 0.33
PKM P14618 1/20 0.33
FDPS P14324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3263348 0.80 TRPA1 (0.36) TRPA1TRPV4TRPV3NPC1PKM
SCHEMBL3264317 0.72 FFAR2 (0.47) TRPA1NPC1PKM
SCHEMBL3266992 0.71 CNR2 (0.35) TRPA1NPC1PKM
SCHEMBL9972900 0.66 ALDH1A1 (0.44) TRPA1
SCHEMBL3266719 0.65 KMT2A (0.35)
SCHEMBL3264475 0.65 TRPA1 (0.33) TRPA1TRPV4
SCHEMBL13537668 0.64 TRPA1 (0.50) TRPA1TRPV4TRPV3
SCHEMBL4026302 0.64 FDPS (0.51) PKMFDPS
SCHEMBL9960985 0.62 NPC1 (0.36) NPC1PKM
SCHEMBL21299172 0.62 FDPS (0.53) PKMFDPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010004390-A1 QUINAZOLINE DIONE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS, S.A. (CH) 2010-01-14 WO claimed
WO-2010004390-A1 QUINAZOLINE DIONE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS, S.A. (CH) 2010-01-14 WO disclosed