SCHEMBL3264376

SCHEMBL3264376

Cc1c(I)c(OC(C)C)nn1-c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 2/20 0.40
NOTUM Q6P988 1/20 0.36
PTGS2 P35354 2/20 0.35
GAA P10253 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
LMNA P02545 2/20 0.35
KMT2A Q03164 3/20 0.35
CACNA2D1 P54289 1/20 0.34
CACNA2D2 Q9NY47 1/20 0.34
P2RY12 Q9H244 1/20 0.34
NR3C1 P04150 1/20 0.34
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3261663 0.85 NPSR1 (0.45) CYP1A2CYP2C19HTTPOLBSMN1; SMN2
SCHEMBL3264878 0.82 CYP1A2 (0.40) CYP1A2CYP2D6CYP2C9CYP2C19HTT
SCHEMBL3264256 0.77 GAA (0.41) CYP1A2CYP2D6CYP2C9CYP2C19HTT
SCHEMBL14151614 0.76 SMN1; SMN2 (0.49) CYP1A2CYP2D6CYP2C9CYP2C19HTT
SCHEMBL3393032 0.75 ATM (0.46) POLBPTGS2GAASMN1; SMN2NPC1
SCHEMBL3386827 0.71 POLB (0.46) POLB
SCHEMBL3390240 0.70 PLK1 (0.39) HTT
SCHEMBL3387671 0.70 POLB (0.69) HTTPOLBPTGS2GAASMN1; SMN2
SCHEMBL3260348 0.70 NPC1 (0.41) POLBNOTUMGAASMN1; SMN2NPC1
SCHEMBL3387939 0.69 SLC5A1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015657-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
WO-2010015657-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
EP-2151433-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed
EP-2151433-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed