SCHEMBL3269983

SCHEMBL3269983

Cc1ccc(Sc2c(OC(N)=O)[nH]c3ccsc23)cc1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
HTT P42858 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GSK3B P49841 1/20 0.34
ADK P55263 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ICAM1 P05362 2/20 0.33
SELE P16581 2/20 0.33
VCAM1 P19320 2/20 0.33
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268889 0.89 MAPK8 (0.32)
SCHEMBL3267982 0.88 MEN1 (0.34) TP53
SCHEMBL3268931 0.88 TUBB4A (0.37) ALDH1A1TDP1
SCHEMBL3268577 0.86 KDR (0.39) ALDH1A1HTTTDP1ICAM1SELE
SCHEMBL3268326 0.85 CCNC (0.33)
SCHEMBL3269102 0.82 PDPK1 (0.36) HTT
SCHEMBL3175728 0.81 PTGS2 (0.41) ALDH1A1HTTL3MBTL1TDP1ICAM1
SCHEMBL3269317 0.81 MEN1 (0.36) GSK3BADKICAM1SELE
SCHEMBL3275434 0.80 EDNRA (0.43) ALDH1A1
SCHEMBL3269989 0.79 KDR (0.39) HTTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed