SCHEMBL3300138

SCHEMBL3300138

CC(C)(C)OC(=O)N(CCN(C(=O)OC(C)(C)C)c1ccc(N2CCc3cc(NS(=O)(=O)c4cc(Cl)cc(Cl)c4)ccc32)nn1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.38
TRIM24 O15164 5/20 0.37
GPR119 Q8TDV5 7/20 0.36
F2 P00734 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRB3 P13945 1/20 0.34
STS P08842 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427429 0.96 HTR6 (0.37) HTR6TRIM24GPR119F2MEN1
SCHEMBL13390149 0.94 GPR119 (0.38) HTR6TRIM24GPR119F2MEN1
SCHEMBL13390156 0.83 GPR119 (0.35) GPR119MEN1KMT2ALMNA
SCHEMBL4553688 0.83 GPR119 (0.35) GPR119MEN1KMT2ALMNATP53
SCHEMBL3305694 0.81 GPR119 (0.34) GPR119
SCHEMBL3295543 0.81 NR1H2 (0.39) GPR119
SCHEMBL3298929 0.81 F2 (0.35) HTR6F2
SCHEMBL13390147 0.80 ADRB2 (0.40) HTR6TRIM24GPR119F2MEN1
SCHEMBL3305215 0.80 GPR119 (0.47) HTR6TRIM24GPR119STS
SCHEMBL3300962 0.79 TRIM24 (0.41) HTR6TRIM24GPR119MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100093703-A1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-15 US disclosed
US-20100093703-A1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-15 US disclosed
WO-2008099000-A2 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093703-A1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS PYGL, PYGM, G6PC1 HTR6 2697/4885TRIM24 3311/4885GPR119 177/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.