SCHEMBL3316808

SCHEMBL3316808

CCCC(=O)NC(Cc1cc(C(F)(F)F)c(N)c(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.48
ITGA2B P08514 5/20 0.48
ACE P12821 5/20 0.41
FAAH O00519 2/20 0.41
ECE1 P42892 1/20 0.40
KIFC1 Q9BW19 2/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
PSMB5 P28074 1/20 0.39
F2R P25116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4479161 0.85 ITGB3 (0.43) ITGB3ITGA2BACEECE1KIFC1
SCHEMBL4479163 0.85 ITGB3 (0.43) ITGB3ITGA2BACEECE1KIFC1
SCHEMBL3314974 0.83 KIFC1 (0.37) ACEECE1KIFC1
SCHEMBL3311174 0.75 ADRB2 (0.43)
SCHEMBL987963 0.75 FAAH (0.64) ITGB3ITGA2BACEFAAHCHRNB2
SCHEMBL265066 0.75 FAAH (0.64) ITGB3ITGA2BACEFAAHCHRNB2
SCHEMBL11793269 0.75 FAAH (0.64) ITGB3ITGA2BACEFAAHCHRNB2
SCHEMBL3310634 0.73 TACR1 (0.44)
SCHEMBL3316803 0.73 TACR1 (0.44)
SCHEMBL3309182 0.73 ACE (0.49) ITGB3ITGA2BACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100113411-A1 Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113411-A1 Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions CALCRL, CALCR, CALCA ITGB3 3048/4885ITGA2B 3269/4885ACE 1176/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.