SCHEMBL3344574

SCHEMBL3344574

COC(=O)c1cc(B(O)O)cnc1OCCc1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
AXL P30530 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
CYP46A1 Q9Y6A2 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HSD17B10 Q99714 2/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ACACB O00763 1/20 0.35
SLC2A1 P11166 1/20 0.35
GCK P35557 1/20 0.35
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345812 0.83 PIM1 (0.43) ALDH1A1KDM4EGLAGAAAXL
SCHEMBL3350903 0.81 ABL1 (0.37) ALDH1A1KDM4EGLAGAATDP1
SCHEMBL3344570 0.77 RORC (0.41) ALDH1A1KDM4EGLAGAAAXL
SCHEMBL3373097 0.76 TBXAS1 (0.47) ALDH1A1KDM4EKMT2A
SCHEMBL3348530 0.76 DGAT1 (0.40) ALDH1A1KDM4EGLAGAAAXL
SCHEMBL3448577 0.72 TSHR (0.44) ALDH1A1TDP1L3MBTL1HSD17B10KMT2A
SCHEMBL19261271 0.70 GAA (0.40) ALDH1A1KDM4EGLAGAACYP46A1
SCHEMBL3346064 0.69 PIM1 (0.51) KMT2ASLC2A1GCKPIM1PIM2
SCHEMBL30601109 0.69 CYP11B1 (0.48) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL29042069 0.69 TSHR (0.42) ALDH1A1KDM4EGLAGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed