SCHEMBL3344704

SCHEMBL3344704

COC(=O)c1cc(C(=O)NCCc2ccccc2)cc(N2CCOC2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 1/20 0.52
RAB9A P51151 11/20 0.52
NPC1 O15118 10/20 0.52
KLF5 Q13887 2/20 0.47
PKM P14618 1/20 0.46
PAX8 Q06710 1/20 0.46
MGLL Q99685 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
HSD17B10 Q99714 1/20 0.42
MAPT P10636 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348715 0.81 KDM1A (0.41) PKMMGLLHSD17B10MAPTLMNA
SCHEMBL3348673 0.76 RAB9A (0.65) KDM5BRAB9ANPC1MGLLHDAC3
SCHEMBL30443816 0.74 KDM1A (0.54) RAB9ANPC1PKMMAPTLMNA
SCHEMBL5853439 0.74 KDM1A (0.54) RAB9ANPC1PKMMAPTLMNA
SCHEMBL8239483 0.74 ALDH1A1 (0.40) RAB9ANPC1PKMMGLLHSD17B10
SCHEMBL1962554 0.73 NOTUM (0.43) PKMMGLLHSD17B10MAPTLMNA
SCHEMBL7272416 0.72 MGLL (0.74) KDM5BRAB9ANPC1MGLLHDAC2
SCHEMBL1015595 0.71 ALDH1A1 (0.52) RAB9ANPC1MGLLHSD17B10SMN1; SMN2
SCHEMBL4747063 0.71 KDM5B (0.56) KDM5BRAB9ANPC1MGLLHDAC3
SCHEMBL4694649 0.70 MCHR1 (0.55) KDM5BRAB9ANPC1MGLLHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042030-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2010-04-15 WO disclosed