SCHEMBL334479

SCHEMBL334479

O=C/C=C/c1ccc(-c2ccccc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.74
TRPA1 O75762 1/20 0.74
LMNA P02545 1/20 0.74
ALOX5 P09917 1/20 0.74
MAPK1 P28482 1/20 0.74
KDM4E B2RXH2 1/20 0.56
MAPT P10636 1/20 0.56
HDAC2 Q92769 2/20 0.50
CA1 P00915 1/20 0.50
MGLL Q99685 1/20 0.50
MAOB P27338 1/20 0.50
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
TP53 P04637 1/20 0.45
XDH P47989 1/20 0.45
CDK4 P11802 3/20 0.44
CCND1 P24385 3/20 0.44
CCNB2 O95067 2/20 0.44
CDK1 P06493 2/20 0.44
CCNB1 P14635 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016496 1.00 ALDH1A1 (0.74) ALDH1A1TRPA1LMNAALOX5MAPK1
Biphenyl SCHEMBL4693704 0.93 ALDH1A1 (0.86) ALDH1A1TRPA1LMNAALOX5MAPK1
SCHEMBL14262692 0.91 ALDH1A1 (0.61) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamaldehyde SCHEMBL28599267 0.86 ALDH1A1 (0.90) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamaldehyde SCHEMBL25267814 0.85 ALDH1A1 (1.00) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamaldehyde SCHEMBL3442 0.85 ALDH1A1 (1.00) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamaldehyde SCHEMBL2203965 0.85 ALDH1A1 (1.00) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamic Aldehyde SCHEMBL1866630 0.85 ALDH1A1 (1.00) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamic Aldehyde SCHEMBL159856 0.85 ALDH1A1 (1.00) ALDH1A1TRPA1LMNAALOX5MAPK1
Cinnamaldehyde SCHEMBL28377500 0.85 ALDH1A1 (1.00) ALDH1A1TRPA1LMNAALOX5MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118388435-A 4-Vinyl dihydrofuran-3, 3 (2H) -disulfonyl difluoro compound, and preparation and application thereof 上海大学 2024-07-26 CN disclosed
EP-3546454-B1 BENZOHETEROCYCLYL ALKYLAMINE COMPOUND AND USE THEREOF UNIV EAST CHINA SCIENCE & TECH (CN) 2023-09-27 EP disclosed
CN-114105993-B Synthesis method of chiral pyrroloimidazole compound 大连理工大学 2023-03-10 CN disclosed
CN-108101826-B Indole-substituted alkylamine compound and application thereof 华东理工大学 2022-05-10 CN disclosed
CN-114105993-A Synthesis method of chiral pyrroloimidazole compound 大连理工大学 2022-03-01 CN disclosed
CN-108117534-B Benzo-oxygenated aliphatic cyclomethylamines 华东理工大学 2021-02-05 CN disclosed
US-10829464-B2 Benzoheterocyclic alkylamine compounds and use thereof EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2020-11-10 US disclosed
CN-108084125-B Benzoheterocyclylalkylamines and their use 华东理工大学 2020-08-18 CN disclosed
US-20190315703-A1 BENZOHETEROCYCLIC ALKYLAMINE COMPOUNDS AND USE THEREOF EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2019-10-17 US disclosed
EP-3546454-A1 BENZOHETEROCYCLYL ALKYLAMINE COMPOUND AND USE THEREOF East China University of Science and Technology (CN) 2019-10-02 EP disclosed
US-20090088454-A1 ANTI-CANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2009-04-02 US disclosed
EP-2019819-A1 NOVEL PEPTIDE DERIVATIVES USEFUL AS ANTIMICROBIAL AGENTS FOR TREATING WOUNDS Neobiotics AB (SE) 2009-02-04 EP disclosed
US-20080255055-A1 Use of Derivatives of Dipeptides for the Manufacture of of a Medicament for the Treamtent of Microbial Infections NEOBIOTICS AB (SE) 2008-10-16 US disclosed
WO-2008124756-A1 COMPOSITIONS AND METHODS FOR TREATING BONE CANCER THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2008-10-16 WO disclosed
US-7427496-B2 Anti-cancer compounds THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2008-09-23 US disclosed
WO-2007129952-A1 NOVEL PEPTIDE DERIVATIVES USEFUL AS ANTIMICROBIAL AGENTS FOR TREATING WOUNDS NEOBIOTICS AB (SE) 2007-11-15 WO disclosed
US-20060183772-A1 To inhibit tumor growth in an animal; to induce apoptosis NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2006-08-17 US disclosed
US-20060116327-A1 Dipeptide derivatives with active agents to formulate one composition to reduce, eliminate more than one microorganism; effect against a broad spectrum of microorganisms; mechanism of action on pathogen may be on a basic level; low probability for developing resistance NEOBIOTICS AB (SE) 2006-06-01 US disclosed
US-5754271-A PHOTOCHROMIC DYES FOR SUNGLASSES AND CONTACT LENSES ESSILOR INTERNATIONAL (COMPAGNIE GENERAL D'OPTIQUE) (FR) 1998-05-19 US disclosed
US-4001130-A DETERGENTS, SUBSTITUTED BUTADIENES HOECHST AKTIENGESELLSCHAFT (DT) 1977-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060116327-A1 Dipeptide derivatives with active agents to formulate one composition to reduce, eliminate more than one microorganism; effect against a broad spectrum of microorganisms; mechanism of action on pathogen may be on a basic level; low probability for developing resistance ARG1, ARGLU1, VIP ALDH1A1 4362/4885TRPA1 1421/4885LMNA 4296/4885
US-20080255055-A1 Use of Derivatives of Dipeptides for the Manufacture of of a Medicament for the Treamtent of Microbial Infections VIP, ARG1, PEPD ALDH1A1 3543/4885TRPA1 1710/4885LMNA 4687/4885
US-10829464-B2 Benzoheterocyclic alkylamine compounds and use thereof AADAC, AAAS, NISCH ALDH1A1 3071/4885TRPA1 732/4885LMNA 1155/4885
US-20190315703-A1 BENZOHETEROCYCLIC ALKYLAMINE COMPOUNDS AND USE THEREOF AADAC, AAAS, NISCH ALDH1A1 3071/4885TRPA1 732/4885LMNA 1155/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.