SCHEMBL3346446

SCHEMBL3346446

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(Cl)cn1)c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.42
CNR1 P21554 4/20 0.40
CNR2 P34972 3/20 0.38
MAPK1 P28482 4/20 0.37
TRPM5 Q9NZQ8 1/20 0.37
KCNH2 Q12809 1/20 0.36
S1PR3 Q99500 1/20 0.35
CHRM4 P08173 1/20 0.35
ADORA2B P29275 1/20 0.35
PARP1 P09874 2/20 0.34
PARP3 Q9Y6F1 1/20 0.34
HTR2B P41595 1/20 0.34
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13364989 0.87 KCNH2 (0.46) ROCK2CNR1KCNH2
SCHEMBL3348197 0.87 KCNH2 (0.46) ROCK2CNR1KCNH2
SCHEMBL13364988 0.87 KCNH2 (0.46) ROCK2CNR1KCNH2
SCHEMBL3349710 0.87 KCNQ3 (0.46) KCNH2
SCHEMBL3346544 0.86 TRPM5 (0.38) ROCK2MAPK1TRPM5KCNH2
SCHEMBL3346452 0.85 KCNH2 (0.48) ROCK2CNR1CNR2MAPK1KCNH2
SCHEMBL3350848 0.84 ROCK2 (0.41) ROCK2MAPK1TRPM5KCNH2
SCHEMBL13365050 0.83 SSTR4 (0.39) ROCK2CNR2MAPK1KCNH2
SCHEMBL3413819 0.83 KCNH2 (0.42) ROCK2CNR2MAPK1KCNH2
SCHEMBL3350804 0.82 MAPK1 (0.41) ROCK2MAPK1KCNH2S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed