SCHEMBL3346461

SCHEMBL3346461

O=C(NCCc1ccccn1)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cn1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.46
MCHR1 Q99705 1/20 0.46
MC4R P32245 2/20 0.45
SCN9A Q15858 3/20 0.44
ALOX5AP P20292 1/20 0.42
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
HTT P42858 1/20 0.41
HSD11B1 P28845 1/20 0.41
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
SCN5A Q14524 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
FPR3 P25089 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346450 0.85 FPR3 (0.48) MC4RALOX5APRAB9AHTTHSD11B1
SCHEMBL3346386 0.80 TAAR1 (0.48) KCNH2MC4RRAB9ANPC1KDM4E
SCHEMBL3346452 0.78 KCNH2 (0.48) KCNH2MC4RKMT2A
SCHEMBL3348201 0.76 CNR1 (0.54) MC4RALOX5APRAB9AHTTHSD11B1
SCHEMBL13365135 0.74 KCNH2 (0.57) KCNH2SCN9A
SCHEMBL3346554 0.72 KCNH2 (0.48) KCNH2MC4R
Hydrochloric Acid SCHEMBL30585928 0.72 HSD11B1 (0.54) ALOX5APRAB9ANPC1HSD11B1KDM4E
Hydrochloric Acid SCHEMBL21640657 0.72 HSD11B1 (0.54) ALOX5APRAB9ANPC1HSD11B1KDM4E
SCHEMBL3349714 0.72 MC4R (0.57) MC4RRAB9ANPC1L3MBTL1ALDH1A1
SCHEMBL3346548 0.71 GPBAR1 (0.39) MC4RRAB9ANPC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed