SCHEMBL3346450

SCHEMBL3346450

O=C(NCCc1ccccn1)[C@@H]1CNC[C@H]1c1ccc(Cl)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR3 P25089 2/20 0.48
CNR1 P21554 1/20 0.48
SMN1; SMN2 Q16637 5/20 0.47
ALOX5AP P20292 1/20 0.44
ALDH1A1 P00352 5/20 0.43
HSD11B1 P28845 1/20 0.43
ROCK2 O75116 1/20 0.42
POLB P06746 1/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
MC4R P32245 1/20 0.41
PKM P14618 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
LMNA P02545 1/20 0.39
FPR2 P25090 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3349714 0.86 MC4R (0.57) CNR1SMN1; SMN2ALDH1A1POLBMC4R
SCHEMBL3348201 0.86 CNR1 (0.54) FPR3CNR1SMN1; SMN2ALOX5APALDH1A1
SCHEMBL3346548 0.85 GPBAR1 (0.39) FPR3ALDH1A1ROCK2KDM4EMC4R
SCHEMBL3346461 0.85 KCNH2 (0.46) FPR3SMN1; SMN2ALOX5APALDH1A1HSD11B1
SCHEMBL3350852 0.83 MC4R (0.37) FPR3ROCK2MC4RMAPT
SCHEMBL3350808 0.82 TAAR1 (0.53) CNR1SMN1; SMN2ALDH1A1POLBKDM4E
SCHEMBL3350885 0.80 TAAR1 (0.47) CNR1ALDH1A1POLBKDM4EMC4R
SCHEMBL3346695 0.77 CNR1 (0.50) CNR1ALDH1A1ROCK2MC4RHTT
SCHEMBL3346446 0.77 ROCK2 (0.42) CNR1ROCK2
Hydrochloric Acid SCHEMBL21640657 0.74 HSD11B1 (0.54) FPR3CNR1SMN1; SMN2ALOX5APALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed