SCHEMBL3347306

SCHEMBL3347306

Cc1cc2nc(CCC#Cc3cccnc3)ccn2n1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 5/20 0.44
CHRNA4 P43681 5/20 0.44
CYP2A6 P11509 4/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2B6 P20813 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP2D6 P10635 3/20 0.40
CYP2E1 P05181 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 2/20 0.39
CYP2C8 P10632 1/20 0.39
GRM5 P41594 7/20 0.39
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345928 0.87 GRM5 (0.36) CYP2C9CYP2C19CYP2D6CYP3A4CYP1A2
SCHEMBL3347641 0.84 GRM5 (0.38) GRM5
SCHEMBL3347525 0.82 CHRNB2 (0.46) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL3346940 0.82 GRM5 (0.42) CYP2D6CYP3A4GRM5
SCHEMBL3345594 0.82 GRM5 (0.40) GRM5
SCHEMBL3347152 0.79 CHRNB2 (0.41) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL3347664 0.79 GRM5 (0.37) GRM5
SCHEMBL3347055 0.79 GRM5 (0.51) CYP1A2GRM5
SCHEMBL3351706 0.78 KDM4E (0.34) GRM5
SCHEMBL3346856 0.78 GRM5 (0.52) CYP2C9CYP2C19CYP2D6CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed