SCHEMBL3348254

SCHEMBL3348254

C#Cc1ccccc1NC(=O)c1ccccc1.c1cn2ncc3c2nc1-3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHB3 P54753 2/20 0.42
IRAK4 Q9NWZ3 6/20 0.40
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 1/20 0.38
CAMKK1 Q8N5S9 1/20 0.38
CAMKK2 Q96RR4 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
TMIGD3 P0DMS9 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.37
KDR P35968 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347002 0.87 MEN1 (0.40) EPHB3IRAK4NPC1RAB9ACAMKK1
SCHEMBL3347267 0.75 TGFBR1 (0.45) EPHB3IRAK4NPC1RAB9ACAMKK1
SCHEMBL3345835 0.75 MAPT (0.40) NPC1RAB9ACAMKK1CAMKK2MEN1
SCHEMBL3346812 0.71 PIM1 (0.40) NPC1RAB9ACAMKK1CAMKK2MEN1
SCHEMBL14897458 0.69 NTRK1 (0.46) EPHB3IRAK4RAB9ATGFBR1
SCHEMBL11225958 0.68 RAB9A (0.62) NPC1RAB9AMEN1KMT2A
SCHEMBL14897663 0.68 ALDH1A1 (0.52) EPHB3ADORA3TMIGD3TGFBR1
SCHEMBL3346996 0.67 MEN1 (0.41) NPC1CYP3A4RAB9ACAMKK1CAMKK2
SCHEMBL16180212 0.66 IRAK4 (0.60) IRAK4IDO1TDO2KDR
SCHEMBL16620804 0.66 KDM4E (0.43) NPC1RAB9ACAMKK1CAMKK2CAMK2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO claimed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed