SCHEMBL3353044

SCHEMBL3353044

O=C(NCCc1cccc(F)c1)[C@@H]1CNC[C@H]1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.46
MC4R P32245 3/20 0.46
CNR1 P21554 1/20 0.45
GLA P06280 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
ROCK2 O75116 2/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
GAA P10253 1/20 0.41
LIPG Q9Y5X9 1/20 0.41
SLC6A2 P23975 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3353041 0.90 CNR1 (0.55) KCNH2MC4RCNR1GLATAAR1
SCHEMBL3346608 0.89 KCNH2 (0.50) KCNH2MC4RCNR1TAAR1ALDH1A1
SCHEMBL3353136 0.88 TAAR1 (0.50) MC4RCNR1GLATAAR1ALDH1A1
SCHEMBL3353235 0.85 ROCK2 (0.49) KCNH2MC4RCNR1ALDH1A1ROCK2
SCHEMBL3353112 0.85 MC4R (0.43) KCNH2MC4RCNR1GLATAAR1
SCHEMBL3346495 0.84 DPP4 (0.50) MC4RCNR1GLATAAR1ALDH1A1
SCHEMBL22179089 0.83 MC4R (0.63) MC4RCNR1GLATAAR1ALDH1A1
SCHEMBL22179092 0.83 MC4R (0.63) MC4RCNR1GLATAAR1ALDH1A1
Hydrochloric Acid SCHEMBL22160598 0.82 MC4R (0.61) MC4RCNR1GLATAAR1ALDH1A1
SCHEMBL2229909 0.79 MC4R (0.63) KCNH2MC4RALDH1A1KMT2AROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed