SCHEMBL336155

SCHEMBL336155

COc1ccc2oc(C(=O)NC(c3ccccc3)C(O)C(=O)Nc3ccc4nc(N)[nH]c4c3)cc2c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 11/20 0.45
TAS1R1 Q7RTX1 11/20 0.45
MAPT P10636 3/20 0.42
RXFP1 Q9HBX9 1/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
TP53 P04637 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 1/20 0.42
BCAT1 P54687 1/20 0.42
MMP2 P08253 1/20 0.41
MMP14 P50281 1/20 0.41
KDR P35968 2/20 0.40
MAOB P27338 1/20 0.40
KDM4E B2RXH2 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335500 0.87 F9 (0.44) RAB9ANPC1SMN1; SMN2KDR
SCHEMBL334843 0.86 KDR (0.45) RAB9ANPC1SMN1; SMN2KDR
SCHEMBL336071 0.86 PYGL (0.45) MAPTRAB9ANPC1TP53TSHR
SCHEMBL335308 0.84 MEN1 (0.44) RXFP1RAB9ANPC1KDR
SCHEMBL335946 0.83 MMP2 (0.38) MAPTRXFP1RAB9ANPC1TP53
SCHEMBL336586 0.81 GRIN1 (0.44) KDR
SCHEMBL335420 0.80 NPC1 (0.46) MAPTRAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL15282285 0.80 ACP1 (0.46) MAPTRAB9ANPC1TP53SMN1; SMN2
SCHEMBL15282212 0.80 ACP1 (0.46) MAPTRAB9ANPC1TP53SMN1; SMN2
SCHEMBL335396 0.79 F7 (0.44) MAPTRAB9ANPC1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US claimed