SCHEMBL3363948

SCHEMBL3363948

Cn1nc2c(-c3ccsc3)cccc2c1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.40
PTGER1 P34995 2/20 0.38
ENPP1 P22413 1/20 0.38
PRKDC P78527 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36
TUBB6 Q9BUF5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3367735 0.86 KDM4E (0.42) ENPP1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3365869 0.84 CYP3A4 (0.40) ENPP1DHODHGABRG2GABRB3GABRA2
SCHEMBL27656681 0.79 TMIGD3 (0.42) GPR35PTGER1ENPP1PRKDCPIK3CD
SCHEMBL3364109 0.79 GABRG2 (0.41) GABRG2GABRB3GABRA2
SCHEMBL3365166 0.78 GABRG2 (0.42) ENPP1DHODHGABRG2GABRB3GABRA2
SCHEMBL3368191 0.77 TUBB4A (0.38) ENPP1PIK3CATUBB4ATUBBTUBA3C
SCHEMBL3367042 0.77 DHODH (0.41) GPR35DHODH
SCHEMBL3368008 0.77 HRH4 (0.43) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL3368049 0.76 DHODH (0.41) DHODH
SCHEMBL3365574 0.75 BRD4 (0.47) GPR35GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed
US-7365211-B2 Heterocyclic GABAA subtype selective receptor modulators ROCHE PALO ALTO LLC (US) 2008-04-29 US disclosed