SCHEMBL3368008

SCHEMBL3368008

Cn1nc2c(-c3ccoc3)cccc2c1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.43
IMPDH2 P12268 2/20 0.41
ELANE P08246 1/20 0.39
TOP2A P11388 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36
TUBB6 Q9BUF5 1/20 0.36
TUBB2B Q9BVA1 1/20 0.36
TUBB1 Q9H4B7 1/20 0.36
GPR84 Q9NQS5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364253 0.86 NR4A2 (0.41) HRH4IMPDH2ELANETOP2ATUBB4A
SCHEMBL3365869 0.84 CYP3A4 (0.40) HRH4SMN1; SMN2HSD17B10ALDH1A1HTT
SCHEMBL3364109 0.79 GABRG2 (0.41) ALDH1A1POLB
SCHEMBL3365166 0.78 GABRG2 (0.42)
SCHEMBL3362490 0.77 HRH4 (0.40) HRH4IMPDH2ELANETOP2ATUBB4A
SCHEMBL3367042 0.77 DHODH (0.41) GAALMNASMN1; SMN2PDE10AUSP2
SCHEMBL3363948 0.77 GPR35 (0.40) TOP2ATUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3368049 0.76 DHODH (0.41)
SCHEMBL3365574 0.75 BRD4 (0.47) GPR84LMNASMN1; SMN2HSD17B10ALDH1A1
SCHEMBL3367559 0.73 PRNP (0.38) HRH4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed
US-7365211-B2 Heterocyclic GABAA subtype selective receptor modulators ROCHE PALO ALTO LLC (US) 2008-04-29 US disclosed