SCHEMBL3368

SCHEMBL3368

Cc1noc(-c2ccc(Br)cc2)c1/C(=C\CCO)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 4/20 0.39
IP6K3 Q96PC2 4/20 0.39
IP6K2 Q9UHH9 4/20 0.39
MCL1 Q07820 2/20 0.37
SLC6A9 P48067 1/20 0.34
PPARD Q03181 2/20 0.34
PPARA Q07869 2/20 0.34
MCHR1 Q99705 1/20 0.33
TRPA1 O75762 1/20 0.33
HPGD P15428 1/20 0.32
BACE1 P56817 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TP53 P04637 1/20 0.32
THRB P10828 1/20 0.32
ACACB O00763 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1736 0.91 NR1H4 (0.35) TRPA1HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL4758 0.87 IP6K1 (0.40) IP6K1IP6K3IP6K2SLC6A9PPARD
SCHEMBL7197 0.84 TBXAS1 (0.39) TRPA1SMN1; SMN2
SCHEMBL7735 0.74 MEN1 (0.34) BACE1MEN1KMT2A
SCHEMBL1633 0.73 NR1H4 (0.33) TRPA1SMN1; SMN2
SCHEMBL1294 0.68 MEN1 (0.34) SMN1; SMN2MEN1KMT2A
SCHEMBL14777413 0.68 IP6K1 (0.40) IP6K1IP6K3IP6K2MCL1PPARD
SCHEMBL13494 0.68 IP6K1 (0.40) IP6K1IP6K3IP6K2MCL1PPARD
SCHEMBL8250811 0.67 PTPN1 (0.36) SMN1; SMN2MEN1KMT2ATP53
SCHEMBL1563 0.66 PTPN1 (0.47) IP6K1IP6K3IP6K2SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed